SCHEMBL7227472

SCHEMBL7227472

CCCNC(=O)c1ccc2c(c1)C(=C(C)Nc1ccc(CN(C)Cc3ccccc3)cc1)C(=O)N2

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 8/20 0.44
SIGMAR1 Q99720 8/20 0.44
ACHE P22303 5/20 0.42
OPRM1 P35372 1/20 0.42
BCHE P06276 1/20 0.41
NAMPT P43490 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.40
GRK5 P34947 1/20 0.40
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7227469 1.00 TMEM97 (0.44) TMEM97SIGMAR1ACHEOPRM1BCHE
SCHEMBL6980870 0.92 SIGMAR1 (0.45) TMEM97SIGMAR1ACHEOPRM1BCHE
SCHEMBL6980866 0.92 SIGMAR1 (0.45) TMEM97SIGMAR1ACHEOPRM1BCHE
SCHEMBL7233906 0.91 NAMPT (0.41) NAMPT
SCHEMBL7233897 0.91 NAMPT (0.41) NAMPT
SCHEMBL7233622 0.89 ACHE (0.44) ACHEBCHENAMPTHDAC1
SCHEMBL7233617 0.89 ACHE (0.44) ACHEBCHENAMPTHDAC1
SCHEMBL7233264 0.88 ACHE (0.46) ACHEBCHENAMPTHDAC1
SCHEMBL7235050 0.86 ACHE (0.45) ACHEBCHENAMPTHDAC1
SCHEMBL7235053 0.86 ACHE (0.45) ACHEBCHENAMPTHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6545035-B1 Having effect on various kinases and cycline/CDK complexes and on the proliferation of various tumour cells. BOEHRINGER INGELHEIM PHARMA KG (DE) 2003-04-08 US disclosed
US-6319918-B1 FOR LYMPHOMA OR SOLID TUMORS TREATMENT BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-11-20 US disclosed