SCHEMBL7229124

SCHEMBL7229124

COC(=O)c1cc(F)cc(N2CCNCC2)c1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 2/20 0.46
CTNNB1 P35222 12/20 0.43
BCL9 O00512 11/20 0.43
TTR P02766 1/20 0.43
CHRM2 P08172 1/20 0.42
CHRM4 P08173 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42
KDR P35968 1/20 0.42
BCL9L Q86UU0 1/20 0.42
MAOB P27338 1/20 0.41
OPRD1 P41143 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL31490556 0.88 ADRB1 (0.51) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL8260952 0.84 TTR (0.46) ADRB1CTNNB1BCL9TTRCHRM2
SCHEMBL23662606 0.83 MRGPRX4 (0.49)
SCHEMBL6505768 0.83 MAOB (0.43) TTRMAOB
SCHEMBL19404305 0.82 TTR (0.56) ADRB1CTNNB1BCL9TTRCHRM2
SCHEMBL19386229 0.82 MAPT (0.46) TTR
SCHEMBL6498944 0.82 ABL1 (0.45) TTR
SCHEMBL19404235 0.81 BCL9 (0.45) CTNNB1BCL9CHRM3OPRD1
SCHEMBL19386237 0.81 CHRNB2 (0.55) ADRB1CTNNB1BCL9TTRCHRM2
SCHEMBL6506081 0.81 ALDH1A1 (0.42) TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6552018-B1 As antitumor agents DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2003-04-22 US disclosed
US-6169086-B1 AN ANTITUMOR AGENT FOR TREATING TUMOR RESISTANT TO 5-FLUOROURACIL TYPE DRUGS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2001-01-02 US disclosed
EP-1022270-A1 PYRAZOLE DERIVATIVES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2000-07-26 EP disclosed