SCHEMBL8260952

SCHEMBL8260952

CC(=O)c1cc(F)cc(N2CCNCC2)c1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.46
ADRB1 P08588 3/20 0.46
CHRM2 P08172 1/20 0.46
CHRM4 P08173 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
MAOB P27338 1/20 0.44
KDR P35968 1/20 0.43
CTNNB1 P35222 11/20 0.42
BCL9 O00512 10/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNA4 P43681 1/20 0.42
BCL9L Q86UU0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19404305 0.86 TTR (0.56) TTRADRB1CHRM2CHRM4CHRM1
SCHEMBL19386237 0.84 CHRNB2 (0.55) TTRADRB1CHRM2CHRM4CHRM1
SCHEMBL7229124 0.84 ADRB1 (0.46) TTRADRB1CHRM2CHRM4CHRM1
SCHEMBL19404236 0.83 CTNNB1 (0.53) CTNNB1BCL9BCL9L
SCHEMBL8259537 0.83 SMN1; SMN2 (0.53) TTRALDH1A1HSD17B10
SCHEMBL6629680 0.81 MAPT (0.49) TTRMAOBALDH1A1TSHR
SCHEMBL3045513 0.79 ADRB1 (0.57) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL12187540 0.79 ADRB1 (0.47) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL26181620 0.78 ALDH1A1 (0.43) ADRB1CHRM2CHRM4CHRM1CHRM3
Hydrochloric Acid SCHEMBL6973293 0.77 ADRB1 (0.55) ADRB1CHRM2CHRM4CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006077424-A1 PHARMACEUTICAL COMPOUNDS ASTEX THERAPEUTICS LIMITED (GB) 2006-07-27 WO disclosed
WO-2006077428-A1 PHARMACEUTICAL COMPOUNDS ASTEX THERAPEUTICS LIMITED (GB) 2006-07-27 WO disclosed
WO-2006077419-A1 PYRAZOLE DERIVATIVES FOR THE INHIBITION OF CDK' S AND GSK' S ASTEX THERAPEUTICS LIMITED (GB) 2006-07-27 WO disclosed