SCHEMBL7229148

SCHEMBL7229148

COC(=O)[C@@H](Cc1ccc(F)cc1)OS(=O)(=O)C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.49
CA7 P43166 3/20 0.49
CA9 Q16790 3/20 0.49
CA14 Q9ULX7 3/20 0.49
NOS2 P35228 5/20 0.43
NOS3 P29474 3/20 0.43
NOS1 P29475 3/20 0.43
PPARG P37231 3/20 0.42
PPARA Q07869 3/20 0.42
TSHR P16473 1/20 0.42
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 1/20 0.40
PTPRB P23467 1/20 0.40
ACE P12821 1/20 0.39
CA2 P00918 1/20 0.39
KDM4E B2RXH2 1/20 0.38
CDK2 P24941 1/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2943750 0.89 MEN1 (0.51) CA12CA7CA9CA14NOS2
SCHEMBL16754029 0.89 MEN1 (0.51) CA12CA7CA9CA14NOS2
SCHEMBL7232459 0.83 PPARG (0.48) CA12CA7CA9CA14PPARG
SCHEMBL8142297 0.76 MEN1 (0.43) CA12CA7CA9CA14PPARG
SCHEMBL7728941 0.76 MEN1 (0.43) CA12CA7CA9CA14PPARG
SCHEMBL7726567 0.76 MEN1 (0.43) CA12CA7CA9CA14PPARG
SCHEMBL10957115 0.75 KMT2A (0.39) CA12CA7CA9CA14PPARG
SCHEMBL8711993 0.75 PPARG (0.44) CA12CA9PPARGPPARAKMT2A
SCHEMBL8711997 0.75 PPARG (0.44) CA12CA9PPARGPPARAKMT2A
SCHEMBL2332745 0.75 CA1 (0.38) CA12CA14MEN1KMT2ACA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230331734-A1 NOVEL SPIROPYRROLIDINE DERIVED ANTIVIRAL AGENTS ENANTA PHARMACEUTICALS, INC. 2023-10-19 US disclosed
US-6514997-B2 Block the activity of picornaviral 3C protease AGOURON PHARMACEUTICALS, INC. 2003-02-04 US disclosed
EP-1252145-A1 ANTIPICORNAVIRAL COMPOUNDS AND COMPOSITIONS, THEIR PHARMACEUTICAL USES, AND MATERIALS FOR THEIR SYNTHESIS AGOURON PHARMACEUTICALS, INC. (US) 2002-10-30 EP disclosed
US-20010047006-A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis AGOURON PHARMACEUTICALS, INC. 2001-11-29 US disclosed
WO-2001040189-A1 ANTIPICORNAVIRAL COMPOUNDS AND COMPOSITIONS, THEIR PHARMACEUTICAL USES, AND MATERIALS FOR THEIR SYNTHESIS AGOURON PHARMACEUTICALS, INC. (US) 2001-06-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230331734-A1 NOVEL SPIROPYRROLIDINE DERIVED ANTIVIRAL AGENTS ACE, PKD1, ACE2 CA12 2916/4885CA7 2636/4885CA9 1685/4885
US-20010047006-A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis RNASE1, SERPINB1, RNASEH1 CA12 1436/4885CA7 1227/4885CA9 1397/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.