SCHEMBL7229708

SCHEMBL7229708

O=C(O)C(CCN1C(=O)c2ccncc2C1=O)COc1ccc(-c2ccccc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 13/20 0.64
MMP9 P14780 13/20 0.64
MMP3 P08254 7/20 0.64
MMP13 P45452 7/20 0.64
MMP1 P03956 3/20 0.64
NPSR1 Q6W5P4 2/20 0.49
TSHR P16473 2/20 0.44
ALDH1A1 P00352 1/20 0.44
HDAC7 Q8WUI4 1/20 0.42
P2RX7 Q99572 1/20 0.41
CYP3A4 P08684 2/20 0.40
CYP2C19 P33261 2/20 0.40
CYP2C9 P11712 1/20 0.40
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
PTPN1 P18031 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7233440 0.90 MMP2 (0.81) MMP2MMP9MMP3MMP13MMP1
SCHEMBL7229104 0.89 MMP2 (0.79) MMP2MMP9MMP3MMP13MMP1
SCHEMBL7225679 0.82 MMP2 (0.80) MMP2MMP9MMP3MMP13MMP1
SCHEMBL7224271 0.81 MMP2 (0.67) MMP2MMP9MMP3MMP13MMP1
SCHEMBL7230149 0.77 MMP2 (0.70) MMP2MMP9MMP3MMP13MMP1
SCHEMBL379517 0.74 NPSR1 (0.48) MMP2MMP9MMP3MMP13MMP1
SCHEMBL7230599 0.72 MMP2 (1.00) MMP2MMP9MMP3MMP13MMP1
SCHEMBL7234102 0.72 MMP2 (0.54) MMP2MMP9MMP3MMP13MMP1
SCHEMBL7224250 0.72 MMP2 (0.81) MMP2MMP9MMP3MMP13MMP1
SCHEMBL7223222 0.71 MMP2 (0.71) MMP2MMP9MMP3MMP13MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6605604-B1 Tumour necrosis factor alpha release inhibitors; efficiency treatment of cancers, rheumatic diseases, arthritis, ulcers, atherosclerosis, asthma LES LABORATOIRES SERVIER (FR) 2003-08-12 US disclosed