SCHEMBL7229822

SCHEMBL7229822

CC(C)N1CCC(N2CC(COc3ccc(CC(NC(=O)OC(C)(C)C)C(=O)O)cc3)OC2=O)CC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.47
ITGA2B P08514 1/20 0.47
PTPN1 P18031 3/20 0.43
MAPK1 P28482 1/20 0.43
YAP1 P46937 1/20 0.42
KMT2A Q03164 3/20 0.41
ATM Q13315 1/20 0.41
HRH2 P25021 1/20 0.40
HRH1 P35367 1/20 0.40
ACE P12821 1/20 0.40
ITGA4 P13612 1/20 0.39
ITGB7 P26010 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
SCN9A Q15858 2/20 0.39
APP P05067 1/20 0.38
ADRB3 P13945 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7228437 0.93 YAP1 (0.42) ITGB3ITGA2BPTPN1MAPK1YAP1
SCHEMBL7229341 0.88 ITGB3 (0.45) ITGB3ITGA2BPTPN1MAPK1YAP1
SCHEMBL7239121 0.83 GRM2 (0.41) ITGB3ITGA2BPTPN1MAPK1ADRB3
SCHEMBL7229825 0.82 ADRB3 (0.39) MAPK1ADRB3
SCHEMBL7236262 0.81 ITGB3 (0.51) ITGB3ITGA2BMAPK1ADRB3
SCHEMBL7237375 0.81 YAP1 (0.44) ITGB3ITGA2BPTPN1MAPK1YAP1
SCHEMBL7231433 0.80 ITGB3 (0.47) ITGB3ITGA2BPTPN1MAPK1YAP1
SCHEMBL7228439 0.80 ADRB3 (0.37) ADRB3
SCHEMBL7238639 0.80 HRH3 (0.38) ADRB3
SCHEMBL7229936 0.77 YAP1 (0.48) ITGB3ITGA2BPTPN1MAPK1YAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602876-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2003-08-05 US disclosed
US-6204280-B1 OXAZOLIDINONE DERIVATIVE, ANTICOAGULANT MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 2001-03-20 US disclosed
EP-0710657-B1 Antagonists of adhesion receptors MERCK PATENT GMBH (DE) 1998-08-26 EP disclosed
EP-0710657-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-08 EP disclosed