SCHEMBL7229341

SCHEMBL7229341

CC(C)(C)OC(=O)NC(=N)N1CCC(N2CC(COc3ccc(CC(NC(=O)OC(C)(C)C)C(=O)O)cc3)OC2=O)CC1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.45
ITGA2B P08514 1/20 0.45
YAP1 P46937 3/20 0.44
PTPN1 P18031 3/20 0.43
MAPK1 P28482 1/20 0.43
KMT2A Q03164 2/20 0.40
HRH2 P25021 1/20 0.40
HRH1 P35367 1/20 0.40
ITGA4 P13612 2/20 0.39
ITGB7 P26010 2/20 0.39
ADRB3 P13945 1/20 0.38
BCL2 P10415 1/20 0.38
ACE P12821 1/20 0.38
HDAC8 Q9BY41 1/20 0.37
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7237375 0.93 YAP1 (0.44) ITGB3ITGA2BYAP1PTPN1MAPK1
SCHEMBL8547886 0.88 ITGB3 (0.46) ITGB3ITGA2BYAP1ADRB3
SCHEMBL7229822 0.88 ITGB3 (0.47) ITGB3ITGA2BYAP1PTPN1MAPK1
SCHEMBL7232013 0.83 ITGB3 (0.40) ITGB3ITGA2BYAP1HRH2HRH1
SCHEMBL7228437 0.81 YAP1 (0.42) ITGB3ITGA2BYAP1PTPN1MAPK1
SCHEMBL7238373 0.78 ITGB3 (0.43) ITGB3ITGA2BYAP1PTPN1MAPK1
SCHEMBL7231433 0.77 ITGB3 (0.47) ITGB3ITGA2BYAP1PTPN1MAPK1
SCHEMBL7228282 0.77 GRM2 (0.47) ITGB3ITGA2BPTPN1
SCHEMBL7229611 0.77 ITGB3 (0.46) ITGB3ITGA2BYAP1PTPN1
SCHEMBL7230723 0.77 ITGB3 (0.42) ITGB3ITGA2BYAP1PTPN1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602876-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2003-08-05 US disclosed
US-6204280-B1 OXAZOLIDINONE DERIVATIVE, ANTICOAGULANT MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 2001-03-20 US disclosed
EP-0710657-B1 Antagonists of adhesion receptors MERCK PATENT GMBH (DE) 1998-08-26 EP disclosed
EP-0710657-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-08 EP disclosed