SCHEMBL7237375

SCHEMBL7237375

COC(=O)C(Cc1ccc(OCC2CN(C3CCN(C(=N)NC(=O)OC(C)(C)C)CC3)C(=O)O2)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
YAP1 P46937 5/20 0.44
HRH2 P25021 1/20 0.38
HRH1 P35367 1/20 0.38
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
KMT2A Q03164 3/20 0.37
MAPK1 P28482 1/20 0.36
PTPN1 P18031 1/20 0.36
ADRB3 P13945 1/20 0.36
GAA P10253 1/20 0.36
MEN1 O00255 1/20 0.36
BCL2 P10415 1/20 0.36
CACNA1B Q00975 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7229341 0.93 ITGB3 (0.45) YAP1HRH2HRH1ITGB3ITGA2B
SCHEMBL7228437 0.88 YAP1 (0.42) YAP1HRH2HRH1ALDH1A1LMNA
SCHEMBL7232013 0.88 ITGB3 (0.40) YAP1HRH2HRH1ITGB3ITGA2B
SCHEMBL8547886 0.84 ITGB3 (0.46) YAP1ITGB3ITGA2BADRB3
SCHEMBL7229822 0.81 ITGB3 (0.47) YAP1HRH2HRH1ITGB3ITGA2B
SCHEMBL7236565 0.78 YAP1 (0.38) YAP1HRH2HRH1ITGB3ITGA2B
SCHEMBL7229145 0.78 YAP1 (0.46) YAP1HRH2HRH1ITGB3ITGA2B
SCHEMBL7229073 0.77 GRM2 (0.45) ITGB3ITGA2B
SCHEMBL7237738 0.77 ITGB3 (0.40) YAP1ITGB3ITGA2BPTPN1
SCHEMBL7235817 0.77 YAP1 (0.39) YAP1HRH2HRH1ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602876-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2003-08-05 US disclosed
US-6204280-B1 OXAZOLIDINONE DERIVATIVE, ANTICOAGULANT MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 2001-03-20 US disclosed
EP-0710657-B1 Antagonists of adhesion receptors MERCK PATENT GMBH (DE) 1998-08-26 EP disclosed
EP-0710657-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-08 EP disclosed