SCHEMBL7230418

SCHEMBL7230418

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(Oc2ccc(NC(=O)C(F)F)cc2)s1

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.32
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
SLC6A3 Q01959 1/20 0.31
HTR3E A5X5Y0 3/20 0.30
HTR3B O95264 3/20 0.30
CHRNA7 P36544 3/20 0.30
HTR3A P46098 3/20 0.30
HTR3D Q70Z44 3/20 0.30
HTR3C Q8WXA8 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7231792 0.89 KMT2A (0.33) KCNH2SLC6A3HTR3EHTR3BCHRNA7
SCHEMBL7231735 0.88 MMP2 (0.36) SMN1; SMN2CHRNA7
SCHEMBL7222908 0.87 EPHX2 (0.34) KDM4ESMN1; SMN2
SCHEMBL7226094 0.85 CHRNA7 (0.42) KCNH2KDM4ELMNASMN1; SMN2HTR3E
SCHEMBL7233323 0.84 ESR1 (0.37) SLC6A3
SCHEMBL7232082 0.84 CXCR2 (0.34) KCNH2LMNASMN1; SMN2SLC6A3HTR3E
SCHEMBL7225066 0.83 SLC6A4 (0.41) KDM4ESLC6A3CHRNA7
SCHEMBL7229845 0.83 SLC6A3 (0.42) SLC6A3
SCHEMBL7225149 0.83 HTR4 (0.37) KDM4ELMNASMN1; SMN2SLC6A3
SCHEMBL7232095 0.83 CHRNA7 (0.34) SLC6A3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed