SCHEMBL7230583

SCHEMBL7230583

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ncc(-c2cc(F)ccn2)o1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FAAH O00519 3/20 0.44
CES1 P23141 1/20 0.44
ACKR3 P25106 9/20 0.40
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
SLC6A3 Q01959 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7232731 0.86 ACKR3 (0.39) FAAHACKR3CA12CA1CA2
SCHEMBL7233239 0.85 CA12 (0.39) ACKR3CA12CA1CA2CA4
SCHEMBL7224879 0.85 AKT1 (0.39) FAAHCES1SLC6A3
SCHEMBL7231889 0.85 FAAH (0.49) FAAH
SCHEMBL7233040 0.84 ACKR3 (0.53) ACKR3
SCHEMBL7234886 0.84 FAAH (0.46) FAAHACKR3CA12CA1CA2
SCHEMBL7225896 0.84 CA12 (0.39) ACKR3CA12CA1CA2CA4
SCHEMBL7226619 0.84 HDAC1 (0.46) FAAHACKR3CA12CA1CA2
SCHEMBL7226238 0.83 ACKR3 (0.35) FAAHCES1ACKR3CA12CA1
SCHEMBL7231627 0.83 CA12 (0.42) ACKR3CA12CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed