SCHEMBL7224879

SCHEMBL7224879

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(-c2cc(F)ccn2)o1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 2/20 0.39
SLC6A3 Q01959 3/20 0.35
MGAM O43451 2/20 0.34
GAA P10253 2/20 0.34
SI P14410 2/20 0.34
MGAM2 Q2M2H8 2/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNA7 P36544 1/20 0.34
CHRNA4 P43681 1/20 0.34
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
TAS1R2 Q8TE23 1/20 0.33
FAAH O00519 1/20 0.33
CES1 P23141 1/20 0.33
KDM1A O60341 1/20 0.33
ULK1 O75385 1/20 0.33
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7230688 0.88 AKT1 (0.44) AKT1SLC6A3MGAMGAASI
SCHEMBL7230583 0.85 FAAH (0.44) SLC6A3FAAHCES1
SCHEMBL7223707 0.85 NPC1 (0.38) AKT1MGAMGAASIMGAM2
SCHEMBL7232903 0.85 SLC6A3 (0.38) AKT1SLC6A3MGAMGAASI
SCHEMBL7224822 0.85 CHRNA7 (0.47) AKT1CHRNB2CHRNA7CHRNA4FAAH
SCHEMBL7230437 0.82 SLC9A1 (0.42) AKT1SLC6A3GAACHRNB2CHRNA4
SCHEMBL7224267 0.82 NPC1 (0.39) AKT1MGAMGAASIMGAM2
SCHEMBL7223511 0.82 S1PR2 (0.48) SLC6A3MGAMGAASIMGAM2
SCHEMBL7231940 0.82 GAA (0.46) SLC6A3MGAMGAASIMGAM2
SCHEMBL7226398 0.82 AKT1 (0.34) AKT1SLC6A3CHRNB2CHRNA7CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed