SCHEMBL7230686

SCHEMBL7230686

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(Sc2cccc(N3CCOCC3)c2)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.35
KMO O15229 1/20 0.35
MAPT P10636 3/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
LMNA P02545 1/20 0.34
CHRNA7 P36544 1/20 0.33
HSD17B1 P14061 2/20 0.33
HSD17B2 P37059 2/20 0.33
F10 P00742 2/20 0.33
RAB9A P51151 2/20 0.33
CASP3 P42574 1/20 0.33
CASP7 P55210 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
NPC1 O15118 1/20 0.33
PLOD2 O00469 1/20 0.32
PLOD3 O60568 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7224240 0.90 F10 (0.35) MAPTMEN1KMT2ALMNAF10
SCHEMBL7231554 0.84 HSD17B1 (0.37) CHRNA7HSD17B1HSD17B2DYRK1ADYRK1B
SCHEMBL7231860 0.84 HSD17B1 (0.48) CHRNA7HSD17B1HSD17B2DYRK1ADYRK1B
SCHEMBL7223520 0.83 CHRNA7 (0.45) CYP2C19KMOCHRNA7DYRK1ADYRK1B
SCHEMBL7232904 0.83 MITF (0.38) MAPTMEN1KMT2ACHRNA7F10
SCHEMBL7225375 0.82 GUSB (0.40) CYP2C19KMOKMT2ANPC1
SCHEMBL7231206 0.82 HSD17B1 (0.37) MAPTCHRNA7HSD17B1HSD17B2RAB9A
SCHEMBL7226168 0.82 HSD17B1 (0.37) HSD17B1HSD17B2F10KDM4E
SCHEMBL7194554 0.82 CHRNA7 (0.52) CHRNA7
SCHEMBL7231965 0.81 CHRNA7 (0.36) CHRNA7HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed