SCHEMBL7225375

SCHEMBL7225375

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(Oc2cccc(N3CCOCC3)c2)s1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GUSB P08236 11/20 0.40
NTRK1 P04629 1/20 0.40
FAAH O00519 3/20 0.36
CYP2C19 P33261 1/20 0.36
KMO O15229 1/20 0.35
OPRK1 P41145 1/20 0.35
NPC1 O15118 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7222867 0.91 ICAM1 (0.38) NTRK1KMT2A
SCHEMBL7231813 0.85 CHRNA7 (0.34) GUSB
SCHEMBL7223520 0.84 CHRNA7 (0.45) CYP2C19KMO
SCHEMBL7223531 0.84 CHRNB4 (0.40) NPC1
SCHEMBL7230230 0.83 GAA (0.38) KMT2A
SCHEMBL7226014 0.83 SLC6A2 (0.41) NPC1
SCHEMBL7225045 0.83 SLC6A3 (0.41)
SCHEMBL7231868 0.83 SLC6A2 (0.41) KMT2A
SCHEMBL7225381 0.82 HTR3E (0.37) NPC1
SCHEMBL7230686 0.82 CYP2C19 (0.35) CYP2C19KMONPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed