SCHEMBL7232006

SCHEMBL7232006

COc1cccc(-c2cnc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)o2)c1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.51
HDAC6 Q9UBN7 4/20 0.51
FAAH O00519 1/20 0.48
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
KMT2A Q03164 2/20 0.44
TP53 P04637 2/20 0.44
HPGD P15428 2/20 0.44
TSHR P16473 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
ALDH1A1 P00352 1/20 0.44
MEN1 O00255 1/20 0.43
VCP P55072 1/20 0.42
PAX8 Q06710 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7232218 0.89 HDAC6 (0.48) HDAC1HDAC6FAAHNPC1RAB9A
SCHEMBL7233865 0.88 HDAC1 (0.49) HDAC1HDAC6GRIN2B
SCHEMBL7231308 0.87 FAAH (0.45) HDAC1HDAC6FAAH
SCHEMBL7223806 0.86 HDAC1 (0.38) HDAC1HDAC6FAAH
SCHEMBL7225821 0.86 HDAC1 (0.50) HDAC1HDAC6
SCHEMBL7234886 0.86 FAAH (0.46) HDAC1HDAC6FAAHPAX8
SCHEMBL7232162 0.86 HDAC1 (0.50) HDAC1HDAC6NPC1RAB9ASMN1; SMN2
SCHEMBL7232700 0.86 FAAH (0.46) HDAC1HDAC6FAAH
SCHEMBL7226103 0.85 SLC9A1 (0.47) HDAC1HDAC6NPC1RAB9AKMT2A
SCHEMBL7073214 0.85 TUBB4A (0.47) HDAC1HDAC6FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed