SCHEMBL7232139

SCHEMBL7232139

Cc1ccccc1Sc1cnc(C(=O)N[C@@H]2C[C@H]3CC[C@@H]2N3)s1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 1/20 0.32
SMYD3 Q9H7B4 1/20 0.32
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A3 Q01959 2/20 0.32
CHRNA1 P02708 1/20 0.32
CHRNG P07510 1/20 0.32
ITGA5 P08648 1/20 0.32
CHRNB1 P11230 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
CHRND Q07001 1/20 0.32
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
ICAM1 P05362 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7233574 0.88 DGAT1 (0.33) USP30SMYD3CHRNB2CHRNA4
SCHEMBL7225735 0.88 CHRNB2 (0.34) SLC6A2SLC6A4SLC6A3CHRNA1CHRNG
SCHEMBL7231098 0.88 HCRTR1 (0.37) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7223713 0.86 CHRNA7 (0.34) USP30CHRNB2CHRNA4HTR3EHTR3B
SCHEMBL7231186 0.84 CHRNA7 (0.33) SLC6A2SLC6A4SLC6A3CHRNA1CHRNG
SCHEMBL7224375 0.84 SLC6A2 (0.38) SMYD3SLC6A2SLC6A4SLC6A3ICAM1
SCHEMBL7225137 0.83 GRM5 (0.35) USP30SLC6A2SLC6A4SLC6A3ICAM1
SCHEMBL7225799 0.82 SLC6A2 (0.36) USP30SMYD3SLC6A2SLC6A4SLC6A3
SCHEMBL7225406 0.81 SLC6A2 (0.33) SLC6A2SLC6A4SLC6A3
SCHEMBL7230414 0.81 USP30 (0.40) USP30SMYD3CHRNB2CHRNA4HTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed