SCHEMBL7234359

SCHEMBL7234359

Nc1ccc(CN2CC=CC2)cc1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.61
LMNA P02545 1/20 0.57
GBA1 P04062 1/20 0.45
GFER P55789 1/20 0.44
CYP3A4 P08684 1/20 0.44
TSHR P16473 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
HRH3 Q9Y5N1 2/20 0.43
LOXL2 Q9Y4K0 1/20 0.42
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
SIGMAR1 Q99720 2/20 0.40
HTR6 P50406 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7231784 0.86 ALDH1A1 (0.56) ALDH1A1LMNAGBA1GFERHRH3
Hydrochloric Acid SCHEMBL10728487 0.85 ALDH1A1 (0.55) ALDH1A1LMNAGBA1GFERHRH3
SCHEMBL6221690 0.83 TAAR1 (0.50) ALDH1A1TDP1HRH3LOXL2MAOB
SCHEMBL10690328 0.81 LMNA (0.80) ALDH1A1LMNAHRH3SIGMAR1HRH4
SCHEMBL3153045 0.77 ALDH1A1 (0.88) ALDH1A1LMNATDP1HRH3HRH4
SCHEMBL54966 0.77 ALDH1A1 (0.96) ALDH1A1LMNAHRH3HRH4
SCHEMBL1241262 0.77 ALDH1A1 (0.57) ALDH1A1LMNAHRH3CYP11B1CYP11B2
SCHEMBL2791022 0.77 MAOA (0.55) ALDH1A1HRH3MAOA
SCHEMBL12082407 0.77 ALDH1A1 (0.59) ALDH1A1LMNAGBA1HRH3
SCHEMBL1639608 0.76 SIGMAR1 (0.65) ALDH1A1LMNACYP3A4TDP1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6545035-B1 Having effect on various kinases and cycline/CDK complexes and on the proliferation of various tumour cells. BOEHRINGER INGELHEIM PHARMA KG (DE) 2003-04-08 US disclosed
US-6319918-B1 FOR LYMPHOMA OR SOLID TUMORS TREATMENT BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-11-20 US disclosed
WO-2000073297-A1 SUBSTITUTED INDOLINONE AS TYROSINE KINASE INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-12-07 WO disclosed
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US disclosed