SCHEMBL7236351

SCHEMBL7236351

COc1ccc(OC)c(-c2ccc(CCC(=O)O)cc2)c1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 15/20 0.65
FFAR4 Q5NUL3 7/20 0.60
ALDH1A1 P00352 1/20 0.53
MAPT P10636 1/20 0.53
HPGD P15428 1/20 0.53
POLB P06746 1/20 0.50
MMEL1 Q495T6 2/20 0.49
MME P08473 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7227936 0.85 FFAR4 (0.67) FFAR1FFAR4MMEL1
SCHEMBL7725124 0.83 FFAR1 (0.58) FFAR1FFAR4MMEL1MME
SCHEMBL14340873 0.82 FFAR1 (0.60) FFAR1FFAR4POLB
SCHEMBL1566761 0.82 FFAR1 (0.73) FFAR1FFAR4ALDH1A1MAPTPOLB
SCHEMBL3677264 0.81 FFAR1 (0.66) FFAR1FFAR4MMEL1MME
SCHEMBL8984877 0.81 FFAR1 (0.57) FFAR1FFAR4
SCHEMBL7235666 0.80 TPH1 (0.69) ALDH1A1MAPTHPGD
SCHEMBL274471 0.80 FFAR1 (0.81) FFAR1FFAR4ALDH1A1POLB
SCHEMBL30792366 0.80 FFAR1 (0.81) FFAR1FFAR4ALDH1A1POLB
SCHEMBL27637469 0.80 FFAR1 (0.59) FFAR1FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6645939-B1 Very late antigen-4 (VLA) integrin antagonists; antiallergens, antiasthmatics, and antiinflammatory agents; multiple sclerosis, autoimmune disease treatment MERCK & CO., INC. 2003-11-11 US disclosed
WO-2000071572-A1 SUBSTITUTED BETA-ALANINE DERIVATIVES AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 2000-11-30 WO disclosed