SCHEMBL7239

SCHEMBL7239

Cc1noc(-c2ccc(Br)cc2)c1C(CO)N[C@H]1CCc2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.38
LMNA P02545 2/20 0.36
TSHR P16473 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PDPK1 O15530 1/20 0.36
KMT2A Q03164 1/20 0.35
MAOA P21397 3/20 0.34
MAOB P27338 3/20 0.34
BCHE P06276 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
ACHE P22303 1/20 0.34
ADRA1A P35348 1/20 0.34
HTR6 P50406 1/20 0.34
BRD4 O60885 3/20 0.34
TAS1R3 Q7RTX0 2/20 0.34
TAS1R1 Q7RTX1 2/20 0.34
TAS1R2 Q8TE23 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7238 0.83 MAOA (0.39) RECQLLMNATSHRALDH1A1HTT
SCHEMBL6762 0.76 P2RX7 (0.50) RECQLLMNATSHRALDH1A1HTT
SCHEMBL7357 0.76 P2RX7 (0.50) RECQLLMNATSHRALDH1A1HTT
SCHEMBL18597749 0.76 P2RX7 (0.50) RECQLLMNATSHRALDH1A1HTT
SCHEMBL6734 0.73 ADRB2 (0.38) LMNATSHRALDH1A1NPSR1KMT2A
SCHEMBL10186261 0.69 PDPK1 (0.49) ALDH1A1HTTPDPK1MAOAMAOB
SCHEMBL7055 0.68 LPAR1 (0.47) RECQLLMNATSHRALDH1A1HTT
SCHEMBL3701232 0.67 LPAR1 (0.48) RECQLLMNATSHRALDH1A1HTT
SCHEMBL2761302 0.67 RAB9A (0.42) LMNAALDH1A1HTTKMT2A
SCHEMBL2836880 0.67 RAB9A (0.42) LMNAALDH1A1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483252-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041694-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed