SCHEMBL7239604

SCHEMBL7239604

Cc1ccnc(O)c1C(N)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT3 Q9NTG7 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
LIMK1 P53667 1/20 0.42
POLB P06746 3/20 0.39
NTRK1 P04629 5/20 0.38
PIM1 P11309 5/20 0.38
NOS3 P29474 2/20 0.38
NOS2 P35228 2/20 0.38
PKMYT1 Q99640 1/20 0.38
ACVR1 Q04771 2/20 0.36
KDM4E B2RXH2 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
CCR1 P32246 1/20 0.34
CCR5 P51681 1/20 0.34
CCR8 P51685 1/20 0.34
KMT2A Q03164 2/20 0.34
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL161321 0.82 SIRT3 (0.46) SIRT3TDP1LIMK1POLBNTRK1
SCHEMBL10766873 0.82 CYP3A4 (0.39) TDP1NOS3NOS2KDM4EL3MBTL1
SCHEMBL31606794 0.82 SIRT3 (0.46) SIRT3TDP1LIMK1POLBNTRK1
Hydrochloric Acid SCHEMBL5012214 0.80 NTRK1 (0.44) SIRT3TDP1LIMK1POLBNTRK1
SCHEMBL29089331 0.80 NTRK1 (0.44) SIRT3TDP1LIMK1POLBNTRK1
Hydrochloric Acid SCHEMBL5012204 0.80 NTRK1 (0.44) SIRT3TDP1LIMK1POLBNTRK1
Ammonia Solution, Strong SCHEMBL27581013 0.80 NTRK1 (0.44) SIRT3TDP1LIMK1POLBNTRK1
SCHEMBL11870742 0.80 SIRT3 (0.44) SIRT3TDP1LIMK1POLBNTRK1
SCHEMBL14917427 0.80 NOS2 (0.52) SIRT3TDP1LIMK1POLBNTRK1
Hydrogen Peroxide SCHEMBL28248198 0.80 NTRK1 (0.48) SIRT3TDP1LIMK1POLBNTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6514997-B2 Block the activity of picornaviral 3C protease AGOURON PHARMACEUTICALS, INC. 2003-02-04 US disclosed
EP-1252145-A1 ANTIPICORNAVIRAL COMPOUNDS AND COMPOSITIONS, THEIR PHARMACEUTICAL USES, AND MATERIALS FOR THEIR SYNTHESIS AGOURON PHARMACEUTICALS, INC. (US) 2002-10-30 EP disclosed
US-20010047006-A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis AGOURON PHARMACEUTICALS, INC. 2001-11-29 US disclosed
WO-2001040189-A1 ANTIPICORNAVIRAL COMPOUNDS AND COMPOSITIONS, THEIR PHARMACEUTICAL USES, AND MATERIALS FOR THEIR SYNTHESIS AGOURON PHARMACEUTICALS, INC. (US) 2001-06-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010047006-A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis RNASE1, SERPINB1, RNASEH1 SIRT3 2116/4885TDP1 1547/4885LIMK1 3951/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.