SCHEMBL7242543

SCHEMBL7242543

CC(NC(=O)OC(C)(C)C)c1cccc(NC(=N)N[N+](=O)[O-])c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.39
HDAC1 Q13547 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
CTSK P43235 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
AURKA O14965 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6547633 0.88 BACE1 (0.42) HDAC4HDAC1ALDH1A1HDAC3HDAC7
SCHEMBL6677825 0.87 PRMT1 (0.39) ALDH1A1CTSKMEN1KMT2ACTSS
SCHEMBL6679014 0.87 HDAC4 (0.41) HDAC4HDAC1ALDH1A1HDAC3HDAC7
SCHEMBL6676268 0.85 CA1 (0.39) HDAC4HDAC1ALDH1A1CTSKBACE1
SCHEMBL6676654 0.83 CTSK (0.43) HDAC4HDAC1HDAC3HDAC7HDAC2
SCHEMBL6676396 0.81 KMT2A (0.40) ALDH1A1MEN1KMT2ALMNAPOLB
SCHEMBL7243182 0.80 AURKA (0.41) HDAC4HDAC1ALDH1A1HDAC3HDAC7
SCHEMBL7247298 0.79 CTSK (0.42) HDAC4HDAC1HDAC3HDAC7HDAC2
SCHEMBL6689701 0.78 RXFP1 (0.42) HDAC1ALDH1A1HDAC3HDAC2HDAC8
SCHEMBL6675639 0.78 ALDH1A1 (0.47) HDAC4HDAC1ALDH1A1HDAC3HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed