SCHEMBL7243182

SCHEMBL7243182

CC(NC(=O)OC(C)(C)C)c1cccc(NC(N)=N[N+](=O)[O-])c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.41
RPS6KB1 P23443 1/20 0.41
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
CTSK P43235 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 2/20 0.37
MAPT P10636 2/20 0.37
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6547640 0.88 PPARG (0.39) AURKARPS6KB1GRIN2DGRIN3BGRIN1
SCHEMBL6679019 0.87 HDAC4 (0.39) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6676274 0.85 CA2 (0.41) AURKARPS6KB1GRIN2DGRIN3BGRIN1
SCHEMBL6676280 0.82 GRIN2D (0.39) AURKARPS6KB1GRIN2DGRIN3BGRIN1
SCHEMBL6675639 0.81 ALDH1A1 (0.47) AURKARPS6KB1MEN1KMT2ACTSK
SCHEMBL6676180 0.81 SIGMAR1 (0.47) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7242543 0.80 HDAC4 (0.39) AURKARPS6KB1MEN1KMT2ACTSK
SCHEMBL6689704 0.79 RXFP1 (0.41) MEN1KMT2ASMN1; SMN2LMNAHTT
SCHEMBL6675007 0.78 GRIN2D (0.49) AURKARPS6KB1GRIN2DGRIN3BGRIN1
SCHEMBL6679740 0.78 AURKA (0.46) AURKARPS6KB1GRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed