SCHEMBL7243105

SCHEMBL7243105

C#CCNC(=N)Nc1cccc(CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
BACE1 P56817 5/20 0.39
KCNQ4 P56696 1/20 0.36
KCNQ5 Q9NR82 1/20 0.36
ACHE P22303 3/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
GRM2 Q14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6678027 0.88 BACE1 (0.40) HDAC3HDAC1HDAC2HDAC10HDAC8
SCHEMBL6679163 0.86 HDAC1 (0.41) HDAC3HDAC1HDAC2BACE1CA1
SCHEMBL6690431 0.85 BACE1 (0.41) BACE1PDK1PDK2PDK3PDK4
SCHEMBL6676782 0.81 BACE1 (0.41) HDAC3MAOAMAOBHDAC1HDAC2
SCHEMBL7243106 0.79 SIGMAR1 (0.39) HDAC3MAOAMAOBHDAC1HDAC2
SCHEMBL6677585 0.79 BACE1 (0.40) HDAC3HDAC1HDAC2BACE1CA1
SCHEMBL6674963 0.78 GLS (0.40) BACE1ACHEPDK1PDK2PDK3
SCHEMBL6677790 0.78 ALDH1A1 (0.47) BACE1ACHEPDK1PDK2PDK3
SCHEMBL6690435 0.76 NOS3 (0.53) BACE1GRM2
SCHEMBL6674967 0.75 GRM2 (0.38) HDAC3HDAC1HDAC2HDAC10HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed