SCHEMBL7243296

SCHEMBL7243296

COc1cc(N)c(S(N)(=O)=O)cc1OC

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.75
CA2 P00918 8/20 0.48
CA1 P00915 7/20 0.48
CA12 O43570 6/20 0.48
CA9 Q16790 6/20 0.48
CA4 P22748 3/20 0.48
CA6 P23280 2/20 0.48
CA5A P35218 2/20 0.48
CA7 P43166 2/20 0.48
CA14 Q9ULX7 2/20 0.48
CA5B Q9Y2D0 2/20 0.48
CA3 P07451 1/20 0.48
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.42
POLB P06746 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
NPC1 O15118 1/20 0.41
P2RX3 P56373 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9645148 0.90 PKM (0.79) PKMCA2CA1CA12CA9
SCHEMBL30068292 0.86 PKM (1.00) PKMCA2CA1CA12CA9
SCHEMBL8777777 0.86 PKM (1.00) PKMCA2CA1CA12CA9
SCHEMBL2777269 0.85 CA12 (0.61) PKMCA2CA1CA12CA9
SCHEMBL3782589 0.85 PKM (0.61) PKMCA2CA1CA12CA9
SCHEMBL7242421 0.85 PKM (0.61) PKMCA2CA1CA12CA9
SCHEMBL17774552 0.82 CA2 (0.65) PKMCA2CA1CA12CA9
SCHEMBL2914715 0.82 PKM (0.56) PKMCA2CA1KDM4EALDH1A1
SCHEMBL9646206 0.81 PKM (0.60) PKMCA2CA1CA12CA9
SCHEMBL10721933 0.81 PKM (0.56) PKMCA2CA1CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1147494-C Novel benzodiazine compound, its preparation method and medicine composition containing them ɪά��ʵ���� 2004-04-28 CN disclosed
US-6635635-B2 5,5-dioxo-2,3,3a,4-tetrahydro-1 H-pyrrolo(2,1-c)(1,2,4)-benzothiadiazin-7-ol, for example; nervous system disorders; alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid (AMPA) modulators LES LABORATOIRES SERVIER (FR) 2003-10-21 US disclosed
US-20020037894-A1 Benzothiadiazine compounds ADIR ET COMPAGNIE (FR) 2002-03-28 US disclosed
CN-1341599-A Novel benzodiazine compound, its preparation method and medicine composition containing them LAB SEUWILL (FR) 2002-03-27 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020037894-A1 Benzothiadiazine compounds HCAR1, GLRA1, HCAR2 PKM 2104/4885CA2 1488/4885CA1 1650/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.