SCHEMBL7244266

SCHEMBL7244266

Cc1c(Br)ccc2c1N(Cc1ccc(S(=O)(=O)N(C)C)cc1)C(=O)C2=O

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARK7 Q99497 3/20 0.50
MAPT P10636 2/20 0.47
TP53 P04637 1/20 0.47
CA12 O43570 9/20 0.44
CA1 P00915 9/20 0.44
CA2 P00918 9/20 0.44
CA9 Q16790 9/20 0.44
ACHE P22303 2/20 0.43
CHRM5 P08912 1/20 0.43
ALDH1A1 P00352 3/20 0.40
ALDH3A1 P30838 2/20 0.40
CA7 P43166 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7245333 0.80 ACHE (0.56) PARK7MAPTTP53CA12CA1
SCHEMBL7245471 0.79 CA12 (0.39) PARK7MAPTCA12CA1CA2
SCHEMBL7243578 0.76 CTRB1 (0.49) PARK7MAPTTP53ACHECHRM5
SCHEMBL17165877 0.73 CYP1B1 (0.49) PARK7MAPTTP53ACHECHRM5
SCHEMBL7252676 0.73 NAMPT (0.40) MAPTCA12CA1CA2CA9
SCHEMBL4908758 0.69 CA1 (0.70) CA12CA1CA2CA9ALDH1A1
SCHEMBL4736390 0.67 PARK7 (1.00) PARK7MAPTTP53CA12CA1
SCHEMBL7245612 0.66 HDAC1 (0.40) CA12CA1CA2CA9ACHE
SCHEMBL7248699 0.66 MAPT (0.42) MAPTCA12CA1CA2CA9
SCHEMBL30774299 0.65 PARK7 (0.82) PARK7MAPTTP53ACHECHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6586447-B1 3,3-disubstituted-oxindole derivatives useful as anticancer agents PFIZER INC 2003-07-01 US disclosed