SCHEMBL7250996

SCHEMBL7250996

COC(=O)C(N)Cc1ccc(OC)cc1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.59
SLC6A4 P31645 1/20 0.58
CYP1A2 P05177 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C19 P33261 1/20 0.54
ALDH1A1 P00352 1/20 0.53
ACACB O00763 1/20 0.51
KIF11 P52732 1/20 0.51
TPH1 P17752 2/20 0.50
HTT P42858 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
DPP4 P27487 1/20 0.49
FAP Q12884 1/20 0.49
DPP8 Q6V1X1 1/20 0.49
DPP9 Q86TI2 1/20 0.49
DPP7 Q9UHL4 1/20 0.49
F2RL1 P55085 1/20 0.49
PTGS2 P35354 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1309076 1.00 LDHA (0.59) LDHASLC6A4CYP1A2CYP2D6CYP2C19
SCHEMBL1311287 1.00 LDHA (0.59) LDHASLC6A4CYP1A2CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL5934842 0.98 LDHA (0.57) LDHASLC6A4CYP1A2CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL7301098 0.98 LDHA (0.57) LDHASLC6A4CYP1A2CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL5934840 0.98 LDHA (0.57) LDHASLC6A4CYP1A2CYP2D6CYP2C19
Iodide SCHEMBL28191565 0.97 LDHA (0.56) LDHASLC6A4CYP1A2CYP2D6CYP2C19
Bromide SCHEMBL28190903 0.97 LDHA (0.56) LDHASLC6A4CYP1A2CYP2D6CYP2C19
SCHEMBL539240 0.95 LDHA (0.54) LDHASLC6A4CYP1A2CYP2D6CYP2C19
SCHEMBL539241 0.95 LDHA (0.54) LDHASLC6A4CYP1A2CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL540603 0.94 TPH1 (0.54) LDHASLC6A4CYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109251163-B Resolution method of indoline-2-formic acid compound and intermediate thereof 江苏永达药业有限公司 2022-12-27 CN claimed
CN-109251163-A A kind of method for splitting of indoline -2- formic acid compound and wherein mesosome 江苏永达药业有限公司 2019-01-22 CN claimed
WO-2025032242-A1 COMPOUNDS AND USES UNIVERSITEIT LEIDEN (NL) 2025-02-13 WO disclosed
CN-109251163-B Resolution method of indoline-2-formic acid compound and intermediate thereof 江苏永达药业有限公司 2022-12-27 CN disclosed
CN-113692401-A Process for producing aromatic amino acid derivative 中外制药株式会社 2021-11-23 CN disclosed
US-11040939-B1 N-transfer reagent and method for preparing the same and its application NATIONAL CHENG KUNG UNIVERSITY (TW) 2021-06-22 US disclosed
WO-2020189540-A1 METHOD FOR PREPARING AROMATIC AMINO ACID DERIVATIVE 中外製薬株式会社 2020-09-24 WO disclosed
CN-109251163-A A kind of method for splitting of indoline -2- formic acid compound and wherein mesosome 江苏永达药业有限公司 2019-01-22 CN disclosed
CN-104860924-B Melanocortin-4 receptor modulators prepare their method and its purposes in human medicine and cosmetics 盖尔德马研究及发展公司 2018-10-09 CN disclosed
CN-104387372-B Oxo azetidine derivatives, preparation method and its purposes in human medical and cosmetics 盖尔德马研究及发展公司 2018-06-26 CN disclosed
CN-108164583-A Proteasome inhibitor and its application 珠海诺贝尔国际生物医药研究院有限公司 2018-06-15 CN disclosed
US-8080576-B2 Compounds for enzyme inhibition ONYX THERAPEUTICS, INC. (US) 2011-12-20 US disclosed
US-8080545-B2 Compounds for enzyme inhibition ONYX THERAPEUTICS, INC. (US) 2011-12-20 US disclosed
US-20100144649-A1 COMPOUNDS FOR ENZYME INHIBITION ONYX THERAPEUTICS, INC. (US) 2010-06-10 US disclosed
US-20100144648-A1 COMPOUNDS FOR ENZYME INHIBITION ONYX THERAPEUTICS, INC. (US) 2010-06-10 US disclosed
US-6610731-B2 Antiinflammatory BRISTOL-MYERS SQUIBB COMPANY 2003-08-26 US disclosed
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US disclosed
CN-1272841-A Novel lactam metalloprotease inhibitors DU PONT PHARM CO (US) 2000-11-08 CN disclosed
WO-1989010751-A1 FUNCTIONALIZED PEPTIDYL AMINODIOLS AND -TRIOLS ABBOTT LABORATORIES (US) 1989-11-16 WO disclosed
EP-0341602-A2 Renin-inhibiting functionalized peptidyl aminodiols and - triols ABBOTT LABORATORIES (US) 1989-11-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11040939-B1 N-transfer reagent and method for preparing the same and its application DNTT, NNMT, NMT1 LDHA 1417/4885SLC6A4 355/4885CYP1A2 547/4885
US-20100144648-A1 COMPOUNDS FOR ENZYME INHIBITION PSME1, PSMB1, PSME3 LDHA 3817/4885SLC6A4 4815/4885CYP1A2 1716/4885
US-20100144649-A1 COMPOUNDS FOR ENZYME INHIBITION PSME1, PSMB1, PSME3 LDHA 3817/4885SLC6A4 4815/4885CYP1A2 1716/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.