SCHEMBL7251900

SCHEMBL7251900

COC(=O)C1=Cc2ccccc2SCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 7/20 0.46
CA9 Q16790 7/20 0.46
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 4/20 0.39
MAPT P10636 2/20 0.38
CYP1A2 P05177 2/20 0.38
POLB P06746 2/20 0.38
CYP2C19 P33261 2/20 0.38
HPGD P15428 2/20 0.38
PLA2G1B P04054 1/20 0.38
ATG4B Q9Y4P1 1/20 0.38
RYR2 Q92736 1/20 0.38
TSHR P16473 2/20 0.37
CA2 P00918 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALOX15 P16050 1/20 0.36
CASP1 P29466 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7247717 0.84 TSHR (0.42) CA12CA9ALDH1A1MAPTCYP1A2
SCHEMBL7250245 0.81 HPGD (0.38) ALDH1A1MAPTHPGDPLA2G1BATG4B
SCHEMBL7221367 0.80 CA12 (0.50) CA12CA9ALDH1A1MAPTCYP1A2
SCHEMBL5211708 0.80 KDM4E (0.39) CA12CA9MEN1KMT2AALDH1A1
SCHEMBL7931723 0.80 POLB (0.41) CA12CA9MEN1KMT2AALDH1A1
SCHEMBL8651466 0.80 ALOX5 (0.38) ALDH1A1MAPTPOLBCYP2C19HPGD
SCHEMBL7385174 0.78 ALDH1A1 (0.42) CA12CA9ALDH1A1MAPTCYP1A2
SCHEMBL7683946 0.76 KDM4E (0.43) CA12CA9MAPTCYP1A2CYP2C19
SCHEMBL7911204 0.74 CA12 (0.50) CA12CA9ALDH1A1HPGDTSHR
SCHEMBL31090834 0.74 CA12 (0.50) CA12CA9ALDH1A1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6566535-B1 Causing an orthohalogenobenzaldehyde or derivative to react with a propanethiol having an electron-attracting group at its 4- position. TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-05-20 US disclosed
EP-1184381-A1 PROCESSES FOR THE PREPARATION OF 2,3-DIHYDROTHIEPINE DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 2002-03-06 EP disclosed
WO-1998055475-A1 GUANIDINE DERIVIATIVES AS INHIBITORS OF NA+/H+ EXCHANGE IN CELLS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-12-10 WO disclosed