SCHEMBL7253554

SCHEMBL7253554

CN(C)CCCn1ccc2ccc(Br)cc21

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.54
HTR2C P28335 3/20 0.54
EGFR P00533 1/20 0.53
HTR1D P28221 8/20 0.51
HTR7 P34969 4/20 0.51
NOS3 P29474 3/20 0.49
NOS1 P29475 3/20 0.49
BPTF Q12830 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7252922 0.91 HTR2A (0.64) HTR2AHTR2CEGFRHTR1DHTR7
SCHEMBL31258100 0.91 HTR2A (0.64) HTR2AHTR2CEGFRHTR1DHTR7
SCHEMBL16741930 0.88 EGFR (0.53) HTR2AHTR2CEGFRHTR7NOS3
SCHEMBL18239699 0.79 HTR7 (0.57) HTR2AHTR2CHTR1DHTR7
SCHEMBL7256513 0.79 HTR7 (0.51) HTR2AHTR2CHTR1DHTR7NOS3
SCHEMBL1049671 0.79 HTR7 (0.51) HTR2AHTR2CHTR7
SCHEMBL6990971 0.78 HTR2A (0.50) HTR2AHTR2CHTR1DNOS3NOS1
SCHEMBL20540198 0.78 HTR2C (0.61) HTR2AHTR2CEGFRHTR1DHTR7
SCHEMBL1121913 0.78 NOS3 (0.53) HTR2AHTR2CHTR1DNOS3NOS1
SCHEMBL3990419 0.78 HTR2C (0.81) HTR2AHTR2CHTR1DNOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6635639-B2 Treatment or diagnosis of central nervous system conditions NPS ALLELIX CORP. (CA) 2003-10-21 US disclosed
US-20020169322-A1 Use of N-alkylamino-heterocylic compounds for the treatment of migraine NPS ALLEXLIX CORP. 2002-11-14 US disclosed
US-6380242-B1 FOR DIAGNOSIS AND THERAPY OF CENTRAL NERVOUS SYSTEM CONDITIONS NPS ALLELIX CORP. (CA) 2002-04-30 US disclosed
EP-1140074-A1 INDOLE AND INDOLIZIDINE DERIVATIVES FOR THE TREATMENT OF MIGRAINE NPS Allelix Corp. (CA) 2001-10-10 EP disclosed
WO-2000038677-A1 INDOLE AND INDOLIZIDINE DERIVATIVES FOR THE TREATMENT OF MIGRAINE ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-07-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020169322-A1 Use of N-alkylamino-heterocylic compounds for the treatment of migraine CNR1, CNR2, KCNH1 HTR2A 425/4885HTR2C 127/4885EGFR 2782/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.