SCHEMBL7254208

SCHEMBL7254208

COc1nc(N)c(Cl)cc1C(C(C)=O)C1CCN(CC(O)C(C)(C)C)CC1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.41
CACNA1I Q9P0X4 1/20 0.41
DRD2 P14416 1/20 0.35
HTR4 Q13639 6/20 0.34
ACHE P22303 3/20 0.34
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
KMT2A Q03164 1/20 0.32
HRH1 P35367 1/20 0.31
CCR3 P51677 1/20 0.31
TLR9 Q9NR96 1/20 0.31
TLR8 Q9NR97 1/20 0.31
TLR7 Q9NYK1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7257990 0.88 KCNH2 (0.41) KCNH2DRD2HTR4ACHE
SCHEMBL7257840 0.87 DRD2 (0.35) KCNH2DRD2HTR4ACHEMEN1
SCHEMBL7254150 0.83 HTR4 (0.45) HTR4ACHEMEN1ALDH1A1CYP2D6
SCHEMBL7254109 0.80 SLC6A2 (0.47) DRD2HTR4ACHE
Hydrochloric Acid SCHEMBL7257864 0.79 SLC6A2 (0.49) DRD2HTR4ACHE
SCHEMBL6329086 0.79 HTR4 (0.52) HTR4ACHEMEN1ALDH1A1CYP2D6
SCHEMBL7259161 0.71 KCNH2 (0.34) KCNH2DRD2TLR9TLR8TLR7
SCHEMBL6328978 0.67 HTR4 (0.54) HTR4ACHEMEN1ALDH1A1CYP2D6
SCHEMBL7259567 0.67 HTR4 (0.42) KCNH2HTR4ACHEMEN1ALDH1A1
SCHEMBL7259062 0.67 HTR4 (0.40) DRD2HTR4ACHEMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003057688-A2 OXO OR OXY-PYRIDINE COMPOUNDS AS 5-HT4 RECEPTOR MODULATORS PFIZER JAPAN INC. (JP) 2003-07-17 WO disclosed