SCHEMBL725528

SCHEMBL725528

O=C1C=Cc2cncnc2C1

nearest known ligand 0.39

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 1/20 0.39
GSK3B P49841 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29427881 1.00 GSK3A (0.39) GSK3AGSK3B
SCHEMBL27998030 0.76
SCHEMBL2771341 0.71
SCHEMBL11349207 0.71 GSK3A (0.37) GSK3AGSK3B
SCHEMBL791362 0.69 GSK3A (0.36) GSK3AGSK3B
SCHEMBL13811980 0.68
SCHEMBL5285232 0.68 GSK3A (0.39) GSK3AGSK3B
SCHEMBL29750384 0.68 GSK3A (0.39) GSK3AGSK3B
SCHEMBL29419946 0.68 GSK3A (0.39) GSK3AGSK3B
SCHEMBL10373645 0.68 GSK3A (0.39) GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 120 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103304492-B The synthetic method of a kind of EGFR inhibitor Dacomitinib HUNAN OUYA BIOLOGICAL CO., LTD. (CN) 2015-12-23 CN claimed
CN-104530063-A Quinazoline and heterocyclic ring compounds, preparing method of compounds, and application of compounds serving as epidermal growth factor receptor inhibitors used for treating cancer BEIJING DALITAI PHARMACEUTICAL TECHNOLOGY CO LTD 2015-04-22 CN claimed
US-20260049089-A1 KRAS INHIBITOR COMPOUND SHANGHAI APEIRON THERAPEUTICS COMPANY LIMITED (CN) 2026-02-19 US disclosed
CN-118324761-A USP inhibitor, preparation method and application thereof 北京华森英诺生物科技有限公司 2024-07-12 CN disclosed
US-20240197891-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING POH DERIVATIVES UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2024-06-20 US disclosed
EP-4374929-A2 METHODS AND DEVICES FOR USING ISOPERILLYL ALCOHOL University of Southern California (US) 2024-05-29 EP disclosed
EP-4323070-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING POH DERIVATIVES UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2024-02-21 EP disclosed
CN-113767106-B Oxazaquinazolin-7 (8H) -ones, preparation method and medical application thereof 劲方医药科技(上海)有限公司 2024-02-20 CN disclosed
WO-2024022471-A1 KRAS INHIBITOR COMPOUND 上海湃隆生物科技有限公司 2024-02-01 WO disclosed
US-20240016800-A1 METHODS OF TREATING NEUROFIBROMATOSIS WITH PERILLYL ALCOHOL UNIVERSITY OF SOUTHERN CALIFORNIA 2024-01-18 US disclosed
EP-4281078-A1 PHARMACEUTICAL COMBINATIONS OF SOS1 INHIBITORS FOR TREATING AND/OR PREVENTING CANCER Lupin Limited (IN) 2023-11-29 EP disclosed
US-20130210877-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING POH DERIVATIVES NEONC TECHNOLOGIES INC. (US) 2013-08-15 US disclosed
US-20130203828-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING POH DERIVATIVES NEO ONCOLOGY INC. (US) 2013-08-08 US disclosed
EP-2609064-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING POH DERIVATIVES Neonc Technologies Inc. (US) 2013-07-03 EP disclosed
CN-102711474-A Quinazoline compounds GLAXOSMITHKLINE LLC 2012-10-03 CN disclosed
WO-2012027693-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING POH DERIVATIVES NEONC TECHNOLOGIES INC. (US) 2012-03-01 WO disclosed
EP-1636236-A1 PYRAZOLO-QUINAZOLINE DERIVATIVES,PROCESS FOR THEIR PREPARATION AND THEIR USE AS KINASE INHIBITORS Pharmacia Italia S.p.A. (IT) 2006-03-22 EP disclosed
WO-2004104007-A1 PYRAZOLO-QUINAZOLINE DERIVATIVES,PROCESS FOR THEIR PREPARATION AND THEIR USE AS KINASE INHIBITORS PHARMACIA ITALIA S.P.A. (IT) 2004-12-02 WO disclosed
WO-1992013092-A1 METHODS OF TRANSCRIPTIONALLY MODULATING EXPRESSION OF HEMATOPOIETIC GROWTH FACTOR GENES ONCOGENE SCIENCE, INC. (US) 1992-08-06 WO disclosed
WO-1992013063-A1 METHODS OF TRANSCRIPTIONALLY MODULATING EXPRESSION OF GROWTH FACTOR GENES AND GROWTH FACTOR RECEPTOR GENES ONCOGENE SCIENCE, INC. (US) 1992-08-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130203828-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING POH DERIVATIVES PLIN3, PLIN5, DOHH GSK3A 1985/4885GSK3B 1727/4885
US-20240197891-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING POH DERIVATIVES PLIN3, PLIN5, PLIN1 GSK3A 2560/4885GSK3B 2702/4885
US-20260049089-A1 KRAS INHIBITOR COMPOUND KRAS, NRAS, HRAS GSK3A 886/4885GSK3B 905/4885
US-20240016800-A1 METHODS OF TREATING NEUROFIBROMATOSIS WITH PERILLYL ALCOHOL PMP22, CHAT, REL GSK3A 4112/4885GSK3B 4441/4885
US-20130210877-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING POH DERIVATIVES PLIN3, PLIN5, DOHH GSK3A 1985/4885GSK3B 1727/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.