SCHEMBL7256183

SCHEMBL7256183

COC(=O)Cc1cc(Br)c(Oc2cc(C(C)C)c(OC)cc2C(=O)c2cc(C)cc(C)c2)c(Br)c1

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.69
THRA P10827 14/20 0.38
THRB P10828 14/20 0.38
ABL1 P00519 1/20 0.35
RIN1 Q13671 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
LMNA P02545 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7053405 0.91 NR3C1 (0.68) NR3C1THRATHRBABL1RIN1
SCHEMBL7253471 0.91 NR3C1 (0.82) NR3C1THRATHRBALOX15TSHR
SCHEMBL5630623 0.91 NR3C1 (0.85) NR3C1THRATHRBABL1RIN1
SCHEMBL7053915 0.89 NR3C1 (0.61) NR3C1THRATHRBLMNA
SCHEMBL7053515 0.88 NR3C1 (0.72) NR3C1THRATHRBLMNA
SCHEMBL7051558 0.88 NR3C1 (0.59) NR3C1THRATHRB
SCHEMBL7050206 0.87 NR3C1 (0.62) NR3C1THRATHRB
SCHEMBL7687151 0.87 NR3C1 (0.62) NR3C1THRATHRB
SCHEMBL7052767 0.87 NR3C1 (0.62) NR3C1THRATHRB
SCHEMBL7681978 0.86 NR3C1 (0.71) NR3C1THRATHRBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030166725-A1 Compounds active at the glucocorticoid receptor KARO BIO AB (SE) 2003-09-04 US disclosed
EP-1265839-A1 COMPOUNDS ACTIVE AT THE GLUCOCORTICOID RECEPTOR KARO BIO AB (SE) 2002-12-18 EP disclosed
WO-2002044120-A1 COMPOUNDS ACTIVE AT THE GLUCOCORTICOID RECEPTOR III KARO BIO AB (SE) 2002-06-06 WO disclosed
WO-2001047859-A1 COMPOUNDS ACTIVE AT THE GLUCOCORTICOID RECEPTOR KARO BIO AB (SE) 2001-07-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030166725-A1 Compounds active at the glucocorticoid receptor NR3C1, NR3C2, GPR119 NR3C1 1/4885THRA 291/4885THRB 167/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.