SCHEMBL7258709

SCHEMBL7258709

Fc1cnc(Nc2ccc3ncccc3c2)nc1-c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.54
ABCB1 P08183 1/20 0.50
ABCC1 P33527 1/20 0.50
ABCG2 Q9UNQ0 1/20 0.50
ULK1 O75385 1/20 0.49
ULK2 Q8IYT8 1/20 0.49
MAPK8 P45983 2/20 0.47
SYK P43405 2/20 0.45
CDK1 P06493 5/20 0.44
PABPC1 P11940 1/20 0.44
AURKA O14965 2/20 0.44
IGF1R P08069 2/20 0.44
GSK3B P49841 2/20 0.44
PLK4 O00444 1/20 0.44
PDPK1 O15530 1/20 0.44
JAK2 O60674 1/20 0.44
PRKD3 O94806 1/20 0.44
MAP4K4 O95819 1/20 0.44
NTRK1 P04629 1/20 0.44
INSR P06213 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6033152 0.83 KDR (0.78) KDRABCB1ABCC1ABCG2MAPK8
SCHEMBL7253189 0.77 MAPT (0.44) SYKSTK17AMEN1NPC1MAPT
SCHEMBL7258541 0.76 SYK (0.58) KDRULK1ULK2MAPK8SYK
SCHEMBL2791886 0.76 ABCB1 (0.61) ABCB1ABCC1ABCG2MAPK8PABPC1
SCHEMBL6210503 0.75 PTK2 (0.54) KDRULK1ULK2MAPK8SYK
SCHEMBL5758552 0.75 NPC1 (0.60) ABCB1ABCC1ABCG2ULK1ULK2
SCHEMBL657592 0.74 SYK (0.76) MAPK8SYKAURKAAURKB
SCHEMBL7258580 0.74 SYK (0.52) KDRULK1ULK2MAPK8SYK
SCHEMBL1011248 0.74 PABPC1 (0.59) ABCB1ABCC1ABCG2MAPK8PABPC1
SCHEMBL4000667 0.73 JAK3 (0.61) KDRMAPK8SYKCDK1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003030909-A1 2- AND 4-AMINOPYRIMIDINES N-SUBSTTITUDED BY A BICYCLIC RING FOR USE AS KINASE INHIBITORS IN THE TREATMENT OF CANCER BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-17 WO disclosed