SCHEMBL7259057

SCHEMBL7259057

COc1ccc(Nc2ccnc(F)c2F)cc1C(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 6/20 0.46
KRAS P01116 2/20 0.40
SOS1 Q07889 2/20 0.40
GAK O14976 9/20 0.39
PTK6 Q13882 1/20 0.38
TGFBR1 P36897 2/20 0.38
RIPK2 O43353 6/20 0.37
COQ8A Q8NI60 6/20 0.37
NLK Q9UBE8 6/20 0.37
EPHB6 O15197 2/20 0.37
ABL1 P00519 2/20 0.37
LCK P06239 2/20 0.37
EPHA1 P21709 2/20 0.37
EPHA8 P29322 2/20 0.37
TXK P42681 1/20 0.37
BMPR1B O00238 1/20 0.37
SRC P12931 1/20 0.37
ACVR1 Q04771 1/20 0.37
MAP2K5 Q13163 1/20 0.37
BCL6 P41182 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7263674 0.74 THRB (0.44) FGFR2
SCHEMBL6692635 0.73 BCL6 (0.41) EGFRBCL6
SCHEMBL7263135 0.72 KRAS (0.33) KRASSOS1
SCHEMBL24942886 0.69 CYP2D6 (0.47)
SCHEMBL26239898 0.68 ALDH1A1 (0.43)
SCHEMBL8119851 0.65 NFE2L2 (0.43)
SCHEMBL10094295 0.65 ABCG2 (0.50)
SCHEMBL15248196 0.65 RPS6KA3 (0.39)
SCHEMBL11984410 0.62 ALDH1A1 (0.58)
SCHEMBL26400628 0.62 KRAS (0.35) KRASSOS1GAK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003094845-A2 PYRIDINE-BASED THYROID RECEPTOR LIGANDS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-11-20 WO disclosed