SCHEMBL7263135

SCHEMBL7263135

COc1ccc(Sc2ccnc(F)c2F)cc1C(C)C

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KRAS P01116 1/20 0.33
SOS1 Q07889 1/20 0.33
PDGFRA P16234 1/20 0.33
KDR P35968 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
GFER P55789 1/20 0.33
P2RX3 P56373 5/20 0.32
P2RX2 Q9UBL9 5/20 0.32
DHFR P00374 2/20 0.32
PTGIR P43119 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
AR P10275 2/20 0.31
MET P08581 1/20 0.31
AXL P30530 1/20 0.31
THRB P10828 1/20 0.30
RORC P51449 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7263674 0.74 THRB (0.44) PDGFRAP2RX3P2RX2THRBRORC
SCHEMBL6690378 0.73 THRB (0.36) KDRPOLBGAAGFERP2RX3
SCHEMBL7259057 0.72 EGFR (0.46) KRASSOS1
SCHEMBL282452 0.71 GAA (0.43) POLBGAAGFERP2RX3P2RX2
SCHEMBL20780317 0.69 GAA (0.47) POLBGAAGFERALDH1A1TSHR
SCHEMBL282378 0.66 AR (0.45) POLBGAAGFERALDH1A1TSHR
SCHEMBL8119851 0.65 NFE2L2 (0.43) POLBGAAGFERP2RX3P2RX2
SCHEMBL6765574 0.65 GAA (0.45) KDRPOLBGAAGFERP2RX3
SCHEMBL15248196 0.65 RPS6KA3 (0.39) TSHRCA1CA2
SCHEMBL7353139 0.64 THRB (0.40) P2RX3P2RX2ALDH1A1THRBRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003094845-A2 PYRIDINE-BASED THYROID RECEPTOR LIGANDS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-11-20 WO disclosed