SCHEMBL7259101

SCHEMBL7259101

CC(C)(C)c1ccncc1-c1ccc(Br)s1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 10/20 0.40
CYP2A6 P11509 10/20 0.40
CYP2B6 P20813 10/20 0.40
CYP2C19 P33261 10/20 0.40
CYP2E1 P05181 9/20 0.40
CYP3A4 P08684 9/20 0.40
CYP2D6 P10635 8/20 0.40
CYP2C9 P11712 8/20 0.40
CYP2C8 P10632 7/20 0.40
MAPT P10636 3/20 0.33
TP53 P04637 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
SNCA P37840 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
CASP1 P29466 1/20 0.33
BLM P54132 1/20 0.33
CASP7 P55210 1/20 0.33
HSD17B10 Q99714 2/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7257140 0.78 CYP1A2 (0.58) CYP1A2CYP2A6CYP2B6CYP2C19CYP2E1
SCHEMBL20576799 0.76 KIF11 (0.38) CYP1A2CYP2A6CYP2B6CYP2C19CYP2E1
SCHEMBL7254285 0.74 CYP2A6 (0.62) CYP1A2CYP2A6CYP2B6CYP2C19CYP2E1
SCHEMBL7259055 0.74 RPS6KA3 (0.43) CYP1A2CYP2A6CYP2B6CYP2C19CYP2E1
SCHEMBL7259061 0.72 CYP2A6 (0.64) CYP1A2CYP2A6CYP2B6CYP2C19CYP2E1
SCHEMBL7253763 0.70 RPS6KA3 (0.37) CYP1A2CYP2A6CYP2B6CYP2C19CYP2E1
SCHEMBL7253747 0.70 CYP2A6 (0.54) CYP1A2CYP2A6CYP2B6CYP2C19CYP2E1
SCHEMBL7253767 0.69 ALOX5 (0.39) CYP3A4MAPTTP53SMN1; SMN2TSHR
SCHEMBL12277223 0.67 SLC22A12 (0.50) CYP1A2CYP2A6CYP2B6CYP2C19CYP2E1
SCHEMBL7253990 0.67 CYP11B2 (0.37) CYP1A2CYP2A6CYP2B6CYP2C19CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003027105-A1 SUBSTITUTED 3-PYRIDYL THIOPHENES AS C17,20 LYASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed