SCHEMBL7263103

SCHEMBL7263103

C[C@H](O)[C@H](CCOc1ccc2ccc(C#N)cc2c1)c1nc(C(N)=O)c[nH]1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADA P00813 1/20 0.46
SLC6A2 P23975 4/20 0.39
SLC6A4 P31645 4/20 0.39
SLC6A3 Q01959 2/20 0.39
HTR3A P46098 1/20 0.39
KCNH2 Q12809 1/20 0.39
SCN9A Q15858 12/20 0.36
FPR2 P25090 2/20 0.36
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
PPARG P37231 1/20 0.33
PPARD Q03181 1/20 0.33
PPARA Q07869 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7263915 0.86 ADA (0.48) ADASCN9AFPR2PPARGPPARD
SCHEMBL7263299 0.86 ADA (0.48) ADAMAPTPPARGPPARDPPARA
SCHEMBL7259601 0.81 ADA (0.44) ADAALDH1A1MAPTPPARGPPARD
SCHEMBL7258942 0.81 ADA (0.43) ADAALDH1A1KDM4E
SCHEMBL7263294 0.79 ADA (0.47) ADAALDH1A1MAPTPPARGPPARA
SCHEMBL5671864 0.77 ADA (0.78) ADA
SCHEMBL7263874 0.75 ADA (0.43) ADAALDH1A1MAPTKDM4ECYP1A2
SCHEMBL7453012 0.74 ADA (0.48) ADAALDH1A1MAPTPPARGPPARD
SCHEMBL7263100 0.73 SCN9A (0.44) ADASLC6A2SLC6A4SLC6A3HTR3A
SCHEMBL7258747 0.73 ADA (0.39) ADASCN9AALDH1A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003006437-A1 IMIDAZOLE DERIVATIVES AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-23 WO disclosed