SCHEMBL7264339

SCHEMBL7264339

C[C@H](O)[C@@H](CCOc1cccc(-c2csc(Cc3ccccc3)n2)c1)NC(=O)c1c[nH]cn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.38
HDAC6 Q9UBN7 2/20 0.38
HDAC1 Q13547 1/20 0.38
ALDH1A1 P00352 5/20 0.37
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
ROCK2 O75116 2/20 0.37
ROCK1 Q13464 2/20 0.37
LMNA P02545 4/20 0.37
RAB9A P51151 3/20 0.37
MAPT P10636 1/20 0.37
ECE1 P42892 1/20 0.37
SMN1; SMN2 Q16637 4/20 0.37
HTT P42858 2/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
NAMPT P43490 1/20 0.37
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
HTR3A P46098 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7263964 0.91 SMN1; SMN2 (0.44) ALDH1A1KMT2AMEN1LMNARAB9A
SCHEMBL7263111 0.90 HDAC8 (0.34) HDAC8HDAC6HDAC1ALDH1A1KMT2A
SCHEMBL7258877 0.82 SMN1; SMN2 (0.40) ALDH1A1KMT2AMEN1ROCK2ROCK1
SCHEMBL7259380 0.81 SMN1; SMN2 (0.39) ALDH1A1KMT2AMEN1ROCK2ROCK1
SCHEMBL7263079 0.80 TP53 (0.46) ALDH1A1ROCK2ROCK1RAB9ASMN1; SMN2
SCHEMBL7258741 0.79 HSD17B1 (0.38) ROCK1RAB9AMAPTSMN1; SMN2GAA
SCHEMBL7259234 0.78 FFAR4 (0.41) ROCK2ROCK1RAB9AMAPTSMN1; SMN2
SCHEMBL7259490 0.78 CNR1 (0.39) ROCK2ROCK1RAB9ASMN1; SMN2HTT
SCHEMBL7263737 0.78 AVPR1B (0.41) RAB9ASMN1; SMN2HTTKDM4ENPC1
SCHEMBL7264346 0.78 ATP4A (0.38) HDAC8HDAC6HDAC1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003006437-A1 IMIDAZOLE DERIVATIVES AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-23 WO claimed
WO-2003006437-A1 IMIDAZOLE DERIVATIVES AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-23 WO disclosed