SCHEMBL7268307

SCHEMBL7268307

CC1(C)C=C(n2ccccc2=O)c2cc([N+](=O)[O-])ccc2O1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
PTPRC P08575 3/20 0.38
S100A4 P26447 2/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
CES1 P23141 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
MAPT P10636 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
POLB P06746 1/20 0.36
CYP3A4 P08684 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CHRM2 P08172 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA2A P08913 1/20 0.36
DRD1 P21728 1/20 0.36
PTGS1 P23219 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085035 0.86 ALDH1A1 (0.38) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL8090151 0.84 ALDH1A1 (0.36) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL8128550 0.84 ALDH1A1 (0.36) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL10695563 0.84 CA9 (0.36) ALDH1A1PTPRCS100A4MEN1KMT2A
SCHEMBL8090699 0.84 ALDH1A1 (0.37) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL9735809 0.84 MEN1 (0.35) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL8090555 0.84 TDP1 (0.37) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL8085305 0.83 ALDH1A1 (0.36) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL8077039 0.83 ALDH1A1 (0.36) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL10697020 0.83 ALDH1A1 (0.36) ALDH1A1PTPRCS100A4BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5391751-A Hypotensive, antiarrhythmia, antiasthmatic agents RED BALLOON INVESTMENT LIMITED (JE) 1995-02-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0346724-A1 Chroman derivates MERCK PATENT GmbH (DE) 1989-12-20 EP disclosed
EP-0273262-A2 Chroman derivatives MERCK PATENT GmbH (DE) 1988-07-06 EP disclosed