SCHEMBL8090699

SCHEMBL8090699

CC1(C)C=C(n2cccc([N+](=O)[O-])c2=O)c2cc([N+](=O)[O-])ccc2O1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
POLB P06746 1/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
TDP1 Q9NUW8 2/20 0.35
CYP3A4 P08684 1/20 0.35
PTPRC P08575 3/20 0.34
S100A4 P26447 2/20 0.34
BCHE P06276 1/20 0.34
ACHE P22303 1/20 0.34
CES1 P23141 1/20 0.34
CASP1 P29466 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10697020 0.88 ALDH1A1 (0.36) ALDH1A1MEN1KMT2ATDP1CYP3A4
SCHEMBL8077039 0.88 ALDH1A1 (0.36) ALDH1A1MEN1KMT2ATDP1CYP3A4
SCHEMBL8085305 0.88 ALDH1A1 (0.36) ALDH1A1MEN1KMT2AGABRA1GABRG2
SCHEMBL7277069 0.86 PDE4A (0.39) POLBTDP1HTTMALT1KDM4E
SCHEMBL8088445 0.86 ADORA3 (0.41) ALDH1A1MEN1KMT2ATDP1CYP3A4
SCHEMBL8085338 0.85 KMT2A (0.38) ALDH1A1MEN1KMT2ACTDSP1GABRA1
SCHEMBL8088352 0.85 KDM4E (0.37) ALDH1A1MEN1KMT2ATDP1CYP3A4
SCHEMBL7268307 0.84 ALDH1A1 (0.39) ALDH1A1POLBMEN1KMT2ANR1H2
SCHEMBL8084793 0.84 CFTR (0.39) ALDH1A1POLBMEN1KMT2AHTT
SCHEMBL8085141 0.83 RECQL (0.44) ALDH1A1POLBTDP1HTTMALT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed