SCHEMBL8090151

SCHEMBL8090151

O=c1ccccn1C1=CC2(CCCC2)Oc2ccc([N+](=O)[O-])cc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
TDP1 Q9NUW8 2/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
PTPRC P08575 3/20 0.35
S100A4 P26447 2/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
CES1 P23141 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MALT1 Q9UDY8 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CYP3A4 P08684 1/20 0.33
LMNA P02545 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8090555 0.99 TDP1 (0.37) ALDH1A1TDP1MAPK1HTTPTPRC
SCHEMBL7268307 0.84 ALDH1A1 (0.39) ALDH1A1TDP1PTPRCS100A4BCHE
SCHEMBL8128550 0.81 ALDH1A1 (0.36) ALDH1A1TDP1HTTPTPRCS100A4
SCHEMBL8084380 0.80 OPRD1 (0.39) MALT1HTR1APDE4D
SCHEMBL8090132 0.79 OPRD1 (0.39) MALT1HTR1APDE4D
SCHEMBL8084291 0.79 OPRD1 (0.39) MALT1HTR1APDE4D
SCHEMBL9735809 0.78 MEN1 (0.35) ALDH1A1TDP1PTPRCS100A4BCHE
SCHEMBL8175110 0.77 OPRD1 (0.39) MALT1LMNANPY5RHTR1APDE4D
SCHEMBL8184423 0.77 MALT1 (0.38) ALDH1A1TDP1MAPK1HTTPTPRC
SCHEMBL8090463 0.76 MALT1 (0.37) ALDH1A1TDP1MAPK1HTTPTPRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed