SCHEMBL7269086

SCHEMBL7269086

CCC(=O)N(C)C1CCN(Cc2ccccc2)CC1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 7/20 0.72
SIGMAR1 Q99720 6/20 0.72
KCNH2 Q12809 2/20 0.67
DRD2 P14416 4/20 0.64
HTR2A P28223 3/20 0.64
HTR2C P28335 3/20 0.64
HTR2B P41595 3/20 0.64
ACHE P22303 1/20 0.59
CHRM3 P20309 5/20 0.59
CHRM2 P08172 4/20 0.59
CCR5 P51681 1/20 0.56
SLC22A1 O15245 1/20 0.55
NR1I2 O75469 1/20 0.55
ABCB1 P08183 1/20 0.55
CHRM1 P11229 1/20 0.55
ADRA2B P18089 1/20 0.55
ADRA2C P18825 1/20 0.55
MAOA P21397 1/20 0.55
DRD4 P21917 1/20 0.55
MAOB P27338 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7278323 0.89 KCNH2 (0.64) OPRM1SIGMAR1KCNH2DRD2HTR2A
SCHEMBL13478882 0.89 KCNH2 (0.67) OPRM1SIGMAR1KCNH2DRD2HTR2A
SCHEMBL5116528 0.89 KCNH2 (0.67) OPRM1SIGMAR1KCNH2DRD2HTR2A
SCHEMBL2845483 0.88 KCNH2 (0.65) OPRM1SIGMAR1KCNH2DRD2HTR2A
SCHEMBL19658765 0.88 OPRM1 (0.56) OPRM1SIGMAR1KCNH2DRD2HTR2A
SCHEMBL784863 0.87 SIGMAR1 (0.68) OPRM1SIGMAR1KCNH2DRD2HTR2A
SCHEMBL9030647 0.86 SIGMAR1 (0.67) OPRM1SIGMAR1KCNH2DRD2HTR2A
SCHEMBL9472071 0.85 SIGMAR1 (0.60) OPRM1SIGMAR1KCNH2DRD2HTR2A
SCHEMBL17533481 0.85 OPRM1 (0.70) OPRM1SIGMAR1KCNH2DRD2HTR2A
SCHEMBL11313073 0.84 SIGMAR1 (0.65) OPRM1SIGMAR1KCNH2DRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5214055-A Analgesics, psychological disorders, anxiolytic agents ADIR ET COMPAGNIE (FR) 1993-05-25 US disclosed
US-5189045-A Antiserotonine agent ADIR ET COMPAGNIE (FR) 1993-02-23 US disclosed
EP-0457686-A1 Novel aminopiperidine, aminopyrrolidine and aminoperhydroazepine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1991-11-21 EP disclosed