SCHEMBL7278323

SCHEMBL7278323

CCCC(=O)N(C)C1CCN(Cc2ccccc2)CC1

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.64
OPRM1 P35372 4/20 0.62
SIGMAR1 Q99720 4/20 0.62
DRD2 P14416 3/20 0.61
HTR2A P28223 3/20 0.61
HTR2C P28335 3/20 0.61
HTR2B P41595 3/20 0.61
ABL1 P00519 1/20 0.57
RIN1 Q13671 1/20 0.57
CHRM2 P08172 4/20 0.57
CHRM3 P20309 4/20 0.57
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
CCR5 P51681 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7269086 0.89 OPRM1 (0.72) KCNH2OPRM1SIGMAR1DRD2HTR2A
SCHEMBL13478882 0.89 KCNH2 (0.67) KCNH2OPRM1SIGMAR1DRD2HTR2A
SCHEMBL5116528 0.86 KCNH2 (0.67) KCNH2OPRM1SIGMAR1DRD2HTR2A
SCHEMBL2845483 0.85 KCNH2 (0.65) KCNH2OPRM1SIGMAR1DRD2HTR2A
SCHEMBL784863 0.85 SIGMAR1 (0.68) KCNH2OPRM1SIGMAR1DRD2HTR2A
SCHEMBL19734931 0.84 OPRM1 (0.58) KCNH2OPRM1SIGMAR1DRD2HTR2A
SCHEMBL9030647 0.83 SIGMAR1 (0.67) KCNH2OPRM1SIGMAR1DRD2HTR2A
SCHEMBL9472071 0.83 SIGMAR1 (0.60) KCNH2OPRM1SIGMAR1DRD2HTR2A
SCHEMBL11313073 0.82 SIGMAR1 (0.65) KCNH2OPRM1SIGMAR1DRD2HTR2A
SCHEMBL27473621 0.82 SIGMAR1 (0.65) KCNH2OPRM1SIGMAR1DRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0457686-B1 Novel aminopiperidine, aminopyrrolidine and aminoperhydroazepine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1994-08-03 EP disclosed
US-5214055-A Analgesics, psychological disorders, anxiolytic agents ADIR ET COMPAGNIE (FR) 1993-05-25 US disclosed
US-5189045-A Antiserotonine agent ADIR ET COMPAGNIE (FR) 1993-02-23 US disclosed
EP-0457686-A1 Novel aminopiperidine, aminopyrrolidine and aminoperhydroazepine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1991-11-21 EP disclosed