SCHEMBL7270880

SCHEMBL7270880

COc1cc(C(C)C#N)cc(OC)c1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.45
DHFR P00374 4/20 0.44
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
MAPT P10636 2/20 0.44
CYP3A4 P08684 1/20 0.43
CA9 Q16790 1/20 0.43
TUBB4A P04350 2/20 0.41
TUBB P07437 2/20 0.41
TUBA3C P0DPH7 2/20 0.41
TUBA1B P68363 2/20 0.41
TUBA4A P68366 2/20 0.41
TUBB4B P68371 2/20 0.41
TUBB3 Q13509 2/20 0.41
TUBB2A Q13885 2/20 0.41
TUBB8 Q3ZCM7 2/20 0.41
TUBA3E Q6PEY2 2/20 0.41
TUBA1A Q71U36 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9039805 0.81 DHFR (0.47) ACHEDHFRPDE4APDE4BPDE4C
SCHEMBL910636 0.80 MAPT (0.47) ACHEDHFRMAPTCYP3A4CA9
SCHEMBL10766570 0.80 MAPT (0.47) ACHEDHFRMAPTCYP3A4CA9
SCHEMBL4036492 0.80 ACHE (0.45) ACHEDHFRMAPTCYP3A4CA9
SCHEMBL4044841 0.80 ACHE (0.45) ACHEDHFRMAPTCYP3A4CA9
SCHEMBL3953279 0.80 ACHE (0.45) ACHEDHFRMAPTCYP3A4CA9
SCHEMBL27819446 0.78 TUBB4A (0.47) ACHEDHFRPDE4APDE4BPDE4C
SCHEMBL9841161 0.78 ACHE (0.55) ACHEPDE4APDE4BPDE4CPDE4D
SCHEMBL27819448 0.78 TUBB4A (0.47) ACHEDHFRPDE4APDE4BPDE4C
Hydrochloric Acid SCHEMBL5742931 0.77 PTGS2 (0.42) ACHEPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0001633-A1 Processes for preparing tri-heterocyclic substituted methanes and their conversion into further intermediates useful in the preparation of pharmacologically active compounds THE WELLCOME FOUNDATION LIMITED (GB) 1979-05-02 EP disclosed