SCHEMBL7270901

SCHEMBL7270901

O=c1[nH]c2ccc(-c3cccnc3)cc2cc1Br

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 7/20 0.52
CYP11B2 P19099 7/20 0.52
MMP2 P08253 1/20 0.52
MMP13 P45452 1/20 0.52
MMP14 P50281 1/20 0.52
CYP19A1 P11511 7/20 0.49
CYP17A1 P05093 2/20 0.49
KDM4E B2RXH2 1/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
FGFR1 P11362 1/20 0.47
IDO1 P14902 1/20 0.46
CLK2 P49760 1/20 0.45
CLK3 P49761 1/20 0.45
DYRK1A Q13627 1/20 0.45
PGR P06401 1/20 0.45
PTGES O14684 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7273923 0.83 AURKA (0.56) CYP11B1CYP11B2MMP2MMP13MMP14
SCHEMBL30516503 0.79 FGFR1 (0.54) CYP11B1CYP11B2CYP19A1CYP17A1FGFR1
Hydrochloric Acid SCHEMBL7273927 0.79 MMP2 (0.54) CYP11B1CYP11B2MMP2MMP13MMP14
SCHEMBL7270988 0.79 RAB9A (0.49) CYP11B1CYP11B2MMP2MMP13MMP14
SCHEMBL4287824 0.78 CYP11B2 (0.57) CYP11B1CYP11B2MMP2MMP13MMP14
SCHEMBL31317820 0.78 CYP19A1 (0.71) CYP11B1CYP11B2MMP2MMP13MMP14
SCHEMBL21812408 0.78 CYP19A1 (0.71) CYP11B1CYP11B2MMP2MMP13MMP14
Hydrochloric Acid SCHEMBL7264278 0.77 CYP11B2 (0.55) CYP11B1CYP11B2MMP2MMP13MMP14
SCHEMBL27671973 0.76 NR4A2 (0.61) CYP11B1CYP11B2MMP2MMP13MMP14
SCHEMBL31475468 0.76 DAO (0.65) KDM4EHPGDHSD17B10CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4710507-A Quinolone inotropic agents PFIZER INC. (US) 1987-12-01 US disclosed
EP-0148623-A2 Quinolone inotropic agents Pfizer Limited (GB) 1985-07-17 EP disclosed