SCHEMBL7271052

SCHEMBL7271052

O=C(OCC1CCCCN1Cc1ccccc1)c1c[nH]c2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.53
ALDH1A1 P00352 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
TSHR P16473 1/20 0.53
THPO P40225 1/20 0.53
HTR4 Q13639 1/20 0.53
PMP22 Q01453 1/20 0.53
HRH3 Q9Y5N1 1/20 0.53
GABRA1 P14867 3/20 0.52
GABRG2 P18507 3/20 0.52
GABRB3 P28472 3/20 0.52
GABRA3 P34903 3/20 0.52
GABRA2 P47869 3/20 0.52
GABRB2 P47870 3/20 0.52
NPC1 O15118 1/20 0.50
MAPT P10636 2/20 0.49
KMT2A Q03164 2/20 0.49
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7278260 0.90 ALDH1A1 (0.54) RAB9AALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL7276029 0.89 RAB9A (0.56) RAB9AALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL7270653 0.86 CYP2D6 (0.56) RAB9AALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL7288972 0.86 GABRA1 (0.47) RAB9AALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL7278463 0.83 CYP2D6 (0.53) RAB9AALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL7269469 0.83 CYP2D6 (0.60) RAB9AALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL7269463 0.83 CYP2D6 (0.60) RAB9AALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL7271039 0.83 CYP2D6 (0.60) RAB9AALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL7277894 0.82 CYP2D6 (0.62) RAB9AALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL7270646 0.80 RAB9A (0.54) RAB9AALDH1A1CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0429984-B1 Indole derivatives NISSHIN FLOUR MILLING CO (JP) 1997-07-23 EP disclosed
US-5124324-A Psychological disorders, 5-hydroxy tryptamine antagonists NISSHIN FLOUR MILLING CO., LTD. (JP) 1992-06-23 US disclosed
EP-0429984-A2 Indole derivatives NISSHIN FLOUR MILLING CO., LTD. (JP) 1991-06-05 EP disclosed