SCHEMBL7272227

SCHEMBL7272227

COc1ccc(CCNC(=O)C(F)(F)F)c2ccc(=O)[nH]c12

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.55
MTNR1A P48039 4/20 0.51
MTNR1B P49286 3/20 0.51
HSD17B10 Q99714 3/20 0.50
TP53 P04637 1/20 0.50
KDM4E B2RXH2 3/20 0.48
TSHR P16473 1/20 0.48
LMNA P02545 1/20 0.46
MAPK1 P28482 1/20 0.46
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C19 P33261 2/20 0.44
ADRB2 P07550 1/20 0.44
DRD2 P14416 1/20 0.44
DRD1 P21728 1/20 0.44
DRD4 P21917 1/20 0.44
DRD3 P35462 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10642833 0.86 HSD17B10 (0.67) ALDH1A1MTNR1AMTNR1BHSD17B10TP53
SCHEMBL10642415 0.81 ALDH1A1 (0.55) ALDH1A1MTNR1AMTNR1BHSD17B10TP53
SCHEMBL22864069 0.80 ALDH1A1 (0.46) ALDH1A1HSD17B10TP53KDM4ETSHR
SCHEMBL9688747 0.78 ALDH1A1 (0.51) ALDH1A1MTNR1AMTNR1BHSD17B10TP53
SCHEMBL11712397 0.76 ADRB2 (0.48) ALDH1A1HSD17B10TP53KDM4ETSHR
Hydrochloric Acid SCHEMBL11035276 0.75 ADRB2 (0.48) ALDH1A1HSD17B10TP53KDM4ETSHR
SCHEMBL7281232 0.75 HTR2A (0.50) ALDH1A1HSD17B10TP53KDM4ELMNA
SCHEMBL10640768 0.74 ADRB2 (0.67) ALDH1A1HSD17B10TP53KDM4ETSHR
SCHEMBL9688803 0.74 MTNR1A (0.44) ALDH1A1MTNR1AMTNR1BHSD17B10TP53
SCHEMBL10641574 0.74 ADRB2 (0.58) ALDH1A1HSD17B10TP53KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0375668-A2 Phenylethylamines, process for their preparation and compositions containing them FISONS plc (GB) 1990-06-27 EP disclosed
US-4868306-A Compounds FISONS PLC (GB) 1989-09-19 US disclosed
US-4791216-A Para ethyl amino phenol pharmaceutical compounds FISONS PLC (GB) 1988-12-13 US disclosed
US-4657929-A Compounds FISONS PLC (GB) 1987-04-14 US disclosed
EP-0142283-A2 Phenylethylamines, process for their preparation and compositions containing them FISONS plc (GB) 1985-05-22 EP disclosed