SCHEMBL7272289

SCHEMBL7272289

O=C(OCC(CO)c1ccccc1)c1cccc(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
RAB9A P51151 2/20 0.48
BCHE P06276 1/20 0.46
ALDH1A1 P00352 2/20 0.45
L3MBTL1 Q9Y468 3/20 0.45
CHRM2 P08172 1/20 0.45
CHRM4 P08173 1/20 0.45
CHRM1 P11229 1/20 0.45
CHRM3 P20309 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
PKM P14618 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MAPK1 P28482 1/20 0.44
GPR139 Q6DWJ6 2/20 0.43
ATM Q13315 1/20 0.43
CASR P41180 1/20 0.42
TRPV1 Q8NER1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7270056 0.89 NPSR1 (0.46) MEN1KMT2ARAB9AALDH1A1CYP1A2
SCHEMBL10640910 0.85 ALDH1A1 (0.49) MEN1KMT2ABCHEALDH1A1L3MBTL1
SCHEMBL7263517 0.84 ADRB2 (0.53) MEN1KMT2ARAB9AALDH1A1L3MBTL1
SCHEMBL7287608 0.84 CYP1A2 (0.44) KMT2AALDH1A1CYP1A2CYP2D6PKM
SCHEMBL10831891 0.83 CYP1A2 (0.41) MEN1KMT2ARAB9AALDH1A1CYP1A2
SCHEMBL7264080 0.82 CYP1A2 (0.45) MEN1KMT2AALDH1A1CYP1A2CYP2D6
SCHEMBL7271252 0.82 GPR139 (0.51) MEN1KMT2ARAB9AL3MBTL1SMN1; SMN2
SCHEMBL10641538 0.80 GPR139 (0.44) MEN1KMT2ARAB9AALDH1A1L3MBTL1
SCHEMBL10635569 0.80 SMN1; SMN2 (0.46) MEN1KMT2ARAB9AALDH1A1L3MBTL1
SCHEMBL10911592 0.78 CES2 (0.45) RAB9AALDH1A1L3MBTL1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0067770-B1 TREATMENT OF MIGRAINE WITH TROPYL BENZOATE DERIVATIVES MERRELL DOW FRANCE ET CIE (FR) 1992-01-15 EP claimed
US-4563465-A ANTISEROTONINE AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1986-01-07 US claimed
EP-0067770-A2 Treatment of migraine with tropyl benzoate derivatives MERRELL DOW FRANCE ET CIE (FR) 1982-12-22 EP claimed
EP-0067770-B1 TREATMENT OF MIGRAINE WITH TROPYL BENZOATE DERIVATIVES MERRELL DOW FRANCE ET CIE (FR) 1992-01-15 EP disclosed
EP-0067770-A2 Treatment of migraine with tropyl benzoate derivatives MERRELL DOW FRANCE ET CIE (FR) 1982-12-22 EP disclosed