SCHEMBL7272801

SCHEMBL7272801

O=[C]CNCCNC(=O)c1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.62
POLB P06746 1/20 0.62
NAAA Q02083 1/20 0.54
GAA P10253 2/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
NPC1 O15118 4/20 0.51
RAB9A P51151 4/20 0.51
EPHX2 P34913 1/20 0.51
PRSS1 P07477 1/20 0.51
CTSG P08311 1/20 0.51
CTRB1 P17538 1/20 0.51
CMA1 P23946 1/20 0.51
HPGD P15428 3/20 0.51
KMT2A Q03164 1/20 0.51
RECQL P46063 1/20 0.50
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18689914 0.85 LMNA (0.69) LMNAPOLBNAAAGAASMN1; SMN2
SCHEMBL237683 0.83 GAA (0.63) LMNAPOLBNAAAGAASMN1; SMN2
SCHEMBL3192014 0.83 LMNA (0.77) LMNAPOLBNAAAGAASMN1; SMN2
SCHEMBL8851577 0.82 LMNA (0.66) LMNAPOLBNAAAGAASMN1; SMN2
SCHEMBL8851817 0.81 DRD2 (0.68) LMNAPOLBNAAAGAASMN1; SMN2
SCHEMBL14067433 0.80 LMNA (0.62) LMNAPOLBNAAAGAASMN1; SMN2
SCHEMBL10784098 0.80 GAA (0.59) LMNAPOLBNAAAGAASMN1; SMN2
SCHEMBL11251484 0.79 LMNA (0.61) LMNAPOLBNAAAGAASMN1; SMN2
SCHEMBL3075535 0.79 LMNA (0.61) LMNAPOLBNAAAGAASMN1; SMN2
SCHEMBL1754794 0.78 LMNA (0.70) LMNAPOLBNAAAGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0049605-B1 SUBSTITUTED ACYL DERIVATIVES OF 1,2,3,4-TETRAHYDROISOQUINOLINE-3-CARBOXYLIC ACIDS, SALTS THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING THE DERIVATIVES OR SALTS, AND THE PRODUCTION OF THE SAME WARNER-LAMBERT COMPANY (US) 1987-03-18 EP disclosed
EP-0037231-B1 SUBSTITUTED ACYL DERIVATIVES OF OCTAHYDRO-1H-INDOLE-2-CARBOXYLIC ACIDS WARNER-LAMBERT COMPANY (US) 1987-01-28 EP disclosed
US-4532342-A N-substituted amino acids as intermediates in the preparation of acyl derivatives of 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acids WARNER-LAMBERT COMPANY (US) 1985-07-30 US disclosed
US-4503043-A HYPOTENSIVES WARNER-LAMBERT COMPANY (US) 1985-03-05 US disclosed
EP-0058567-B1 SUBSTITUTED ACYL DERIVATIVES OF OCTAHYDRO-1H-ISOINDOLE-1-CARBOXYLIC ACIDS AND ESTERS WARNER-LAMBERT COMPANY (US) 1984-07-25 EP disclosed
US-4425355-A HYPOTENSIVE WARNER-LAMBERT COMPANY (US) 1984-01-10 US disclosed
EP-0096157-A2 Substituted acyl derivatives of 1,2,3,4-tetrahydro-6,7-dimethoxy-3-isoquinolinecarboxylic acid WARNER-LAMBERT COMPANY (US) 1983-12-21 EP disclosed
EP-0088342-A1 Substituted acyl derivatives of octahydro-1H-indole-2-carboxylic acids WARNER-LAMBERT COMPANY (US) 1983-09-14 EP disclosed
US-4350704-A HYPOTENSIVE AGENTS WARNER-LAMBERT COMPANY (US) 1982-09-21 US disclosed
US-4344949-A Substituted acyl derivatives of 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acids WARNER-LAMBERT COMPANY (US) 1982-08-17 US disclosed
EP-0049605-A1 Substituted acyl derivatives of 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acids, salts thereof, pharmaceutical compositions containing the derivatives or salts, and the production of the same WARNER-LAMBERT COMPANY (US) 1982-04-14 EP disclosed
EP-0037231-A2 Substituted acyl derivatives of octahydro-1H-indole-2-carboxylic acids WARNER-LAMBERT COMPANY (US) 1981-10-07 EP disclosed