SCHEMBL7272852

SCHEMBL7272852

CC(C)(C)OC(=O)NCCCCCC(=O)NC[C@@H]1C[C@@H](CC(=O)O)C(=O)N1CCc1ccc2ccccc2c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.40
CYP3A4 P08684 1/20 0.40
HDAC1 Q13547 3/20 0.38
HDAC8 Q9BY41 3/20 0.38
HDAC3 O15379 2/20 0.38
GBA1 P04062 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
CACNA1G O43497 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
HDAC2 Q92769 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
DRD2 P14416 1/20 0.36
TLR2 O60603 1/20 0.36
TLR1 Q15399 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7276194 0.92 SIGMAR1 (0.47) SIGMAR1CYP3A4HDAC1HDAC8HDAC3
SCHEMBL7275772 0.91 CYP3A4 (0.39) SIGMAR1CYP3A4HDAC1HDAC8HDAC3
SCHEMBL7273844 0.88 SIGMAR1 (0.51) SIGMAR1CYP3A4HDAC1HDAC8HDAC3
SCHEMBL7275131 0.88 SIGMAR1 (0.51) SIGMAR1CYP3A4HDAC1HDAC8HDAC3
SCHEMBL7274594 0.88 SIGMAR1 (0.51) SIGMAR1CYP3A4HDAC1HDAC8HDAC3
SCHEMBL7274726 0.87 SIGMAR1 (0.51) SIGMAR1CYP3A4HDAC1HDAC8HDAC3
SCHEMBL7275503 0.87 GBA1 (0.40) SIGMAR1CYP3A4HDAC1HDAC8HDAC3
SCHEMBL7274136 0.86 HDAC1 (0.39) HDAC1HDAC8HDAC3HDAC6HDAC2
SCHEMBL7282728 0.85 SIGMAR1 (0.40) SIGMAR1CA1CA2
SCHEMBL7272799 0.85 HDAC1 (0.41) HDAC1HDAC8HDAC3HDAC6HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed