SCHEMBL7275503

SCHEMBL7275503

CC(C)(C)OC(=O)NCCCCCC(=O)NC[C@@H]1C[C@@H](CC(=O)O)C(=O)N1CCc1cccc2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.40
DRD2 P14416 2/20 0.40
NQO2 P16083 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPT P10636 1/20 0.38
SIGMAR1 Q99720 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
CACNA1G O43497 1/20 0.37
TLR7 Q9NYK1 2/20 0.36
TLR8 Q9NR97 1/20 0.36
TLR2 O60603 1/20 0.36
TLR1 Q15399 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7274916 0.91 DRD2 (0.41) GBA1DRD2NQO2CYP3A4MAPT
SCHEMBL7276194 0.89 SIGMAR1 (0.47) GBA1DRD2CYP3A4SIGMAR1HDAC3
SCHEMBL7272983 0.87 GRB2 (0.37) HDAC3HDAC1HDAC8HDAC6
SCHEMBL7272852 0.87 SIGMAR1 (0.40) GBA1DRD2CYP3A4MAPTSIGMAR1
SCHEMBL7275131 0.86 SIGMAR1 (0.51) GBA1CYP3A4SIGMAR1HDAC3HDAC1
SCHEMBL7274594 0.86 SIGMAR1 (0.51) GBA1CYP3A4SIGMAR1HDAC3HDAC1
SCHEMBL7273844 0.86 SIGMAR1 (0.51) GBA1CYP3A4SIGMAR1HDAC3HDAC1
SCHEMBL7274726 0.85 SIGMAR1 (0.51) CYP3A4SIGMAR1HDAC3HDAC1HDAC8
SCHEMBL7283712 0.85 CA12 (0.38) MAPTHDAC3HDAC1HDAC8HDAC6
SCHEMBL7282422 0.84 CYP3A4 (0.47) GBA1CYP3A4MAPTSIGMAR1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed