SCHEMBL7272983

SCHEMBL7272983

N=C(N)NCCCCCC(=O)NC[C@@H]1C[C@@H](CC(=O)O)C(=O)N1CCc1cccc2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRB2 P62993 2/20 0.37
MTNR1A P48039 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA3 P07451 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
EPHX2 P34913 1/20 0.36
CCR4 P51679 2/20 0.35
MC4R P32245 1/20 0.35
MC5R P33032 1/20 0.35
MC3R P41968 1/20 0.35
MC1R Q01726 1/20 0.35
TPSAB1 Q15661 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7283712 0.90 CA12 (0.38) MTNR1ACA12CA1CA2CA3
SCHEMBL7274864 0.88 NAMPT (0.40) MTNR1AITGB3ITGA2BHDAC3HDAC1
SCHEMBL7275503 0.87 GBA1 (0.40) HDAC3HDAC1HDAC8HDAC6
SCHEMBL7274136 0.87 HDAC1 (0.39) MC4RMC5RMC3RMC1RITGB3
SCHEMBL7272690 0.86 NAMPT (0.41) ITGB3ITGA2BHDAC3HDAC1HDAC2
SCHEMBL7284310 0.86 NAMPT (0.41) ITGB3ITGA2BHDAC3HDAC1HDAC2
SCHEMBL7272971 0.86 NAMPT (0.41) ITGB3ITGA2BHDAC3HDAC1HDAC2
SCHEMBL7274469 0.85 LMNA (0.42) ITGB3ITGA2BHDAC3HDAC1HDAC2
SCHEMBL7282847 0.83 HDAC3 (0.41) MTNR1AITGB3ITGA2BHDAC3HDAC4
SCHEMBL7274533 0.82 TSHR (0.40) MTNR1AITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed